Mutations
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5HT1B | 5-HT1B | 3x41 | 138 | TM3 | L | W | thermostabilising | 4IAR, 4IAQ, 7C61, 5V54 |
5HT2B | 5-HT2B | 3x41 | 144 | TM3 | M | W | thermostabilising | 6DS0, 6DRY, 5TVN, 4IB4, 5TUD, 4NC3, 6DRZ, 6DRX |
5HT2C | 5-HT2C | 7x45 | 360 | TM7 | C | N | thermostabilising, receptor-expression | 6BQH, 6BQG |
AA1R | A1 | 159 | ECL2 | N | A | glycosylation-site | 5UEN, 5N2S | |
AA1R | A1 | 2x52 | 57 | TM2 | A | L | thermostabilising | 5N2S |
AA1R | A1 | 3x36 | 91 | TM3 | T | A | thermostabilising | 5N2S |
AA1R | A1 | 5x63 | 205 | TM5 | Y | A | thermostabilising | 5N2S |
AA1R | A1 | 6x37 | 236 | TM6 | L | A | thermostabilising | 5N2S |
AA1R | A1 | 6x41 | 240 | TM6 | L | A | thermostabilising | 5N2S |
AA1R | A1 | 7x41 | 277 | TM7 | T | A | thermostabilising | 5N2S |
AA1R | A1 | 8x64 | 309 | H8 | C | S | palmitoylation-site | 5N2S |
AA2AR | A2A | 2x52 | 54 | TM2 | A | L | thermostabilising | 2YDV, 5IU7, 4UHR, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 4UG2, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 2YDO, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 3x36 | 88 | TM3 | T | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 3x55 | 107 | TM3 | R | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 4x43 | 122 | TM4 | K | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 5x63 | 202 | TM5 | L | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 6x37 | 235 | TM6 | L | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 6x41 | 239 | TM6 | V | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 7x41 | 277 | TM7 | S | A | thermostabilising | 5IU7, 5NM4, 5NM2, 5OLO, 5OLH, 3UZC, 5IUA, 5IU4, 5N2R, 3RFM, 3UZA, 5IU8, 5NLX, 5MZJ, 5OLG, 3REY, 3PWH, 5IUB, 5OM4, 5OLV, 5OM1, 5MZP, 5OLZ |
AA2AR | A2A | 3x39 | 91 | TM3 | S | A | thermostabilising | 5WF6 |
AA2AR | A2A | 154 | ECL2 | N | Q | glycosylation-site | 3VGA, 3VG9 | |
AA2AR | A2A | 154 | ECL2 | N | A | glycosylation-site | 2YDV, 5IU7, 6GDG, 4UHR, 5NM4, 5NM2, 5OLO, 5OLH, 5IUA, 5IU4, 4UG2, 5G53, 5N2R, 5IU8, 5NLX, 5MZJ, 5OLG, 5OM4, 5IUB, 2YDO, 5OLV, 5OM1, 5MZP, 5OLZ | |
AA2AR | A2A | 2x46 | 48 | TM2 | L | A | thermostabilising | 2YDO, 4UG2, 2YDV, 4UHR |
AA2AR | A2A | 2x62 | 65 | TM2 | T | A | thermostabilising | 2YDO, 4UG2, 2YDV, 4UHR |
AA2AR | A2A | 3x37 | 89 | TM3 | Q | A | thermostabilising | 2YDO, 4UG2, 2YDV, 4UHR |
AA2AR | A2A | 2x50 | 52 | TM2 | D | N | thermostabilising | 5WF5 |
ACM1 | M1 | 2 | N-term | N | Q | glycosylation-site | 6OIJ, 6WJC, 5CXV | |
ACM1 | M1 | 12 | N-term | N | Q | glycosylation-site | 6OIJ, 6WJC, 5CXV | |
ACM1 | M1 | 3x37 | 110 | TM3 | N | Q | glycosylation-site | 6OIJ, 6WJC, 5CXV |
ACM2 | M2 | 2 | N-term | N | D | glycosylation-site | 3UON, 4MQS, 4MQT | |
ACM2 | M2 | 3 | N-term | N | D | glycosylation-site | 3UON, 4MQS, 4MQT, 6OIK | |
ACM2 | M2 | 6 | N-term | N | D | glycosylation-site | 7T8X, 6OIK, 7T90, 4MQS, 7T94, 3UON, 7T96, 4MQT | |
ACM2 | M2 | 9 | N-term | N | D | glycosylation-site | 7T8X, 6OIK, 7T90, 4MQS, 7T94, 3UON, 7T96, 4MQT | |
ACM2 | M2 | 373 | ICL3 | A | T | other-effect | 4MQS, 4MQT | |
ACM2 | M2 | 374 | ICL3 | K | R | other-effect | 4MQS, 4MQT | |
ADRB1 | β1 | 1x59 | 68 | TM1 | R | S | thermostabilising | 2Y00, 6H7J, 6H7O, 6H7N, 6IBL, 2Y02, 5F8U, 2YCZ, 3ZPQ, 2Y03, 2Y04, 4AMJ, 4AMI, 2Y01, 2VT4, 2YCY, 4GPO, 2YCX, 6H7M, 5A8E, 3ZPR, 4BVN, 2YCW, 6H7L |
ADRB1 | β1 | 2x53 | 90 | TM2 | M | V | thermostabilising | 2Y00, 6H7J, 6H7O, 6H7N, 6IBL, 2Y02, 5F8U, 2YCZ, 3ZPQ, 2Y03, 2Y04, 4AMJ, 4AMI, 2Y01, 2VT4, 2YCY, 4GPO, 2YCX, 6H7M, 5A8E, 3ZPR, 4BVN, 6TKO, 2YCW, 6H7L |
ADRB1 | β1 | 3x27 | 116 | TM3 | C | L | receptor-expression | 2Y00, 6H7J, 6H7O, 6H7N, 6IBL, 2Y02, 5F8U, 2YCZ, 3ZPQ, 2Y03, 2Y04, 4AMJ, 4AMI, 2Y01, 2VT4, 2YCY, 4GPO, 2YCX, 6H7M, 5A8E, 3ZPR, 4BVN, 6TKO, 2YCW, 6H7L |
ADRB1 | β1 | 7x36 | 327 | TM7 | F | A | thermostabilising | 2Y00, 6H7J, 6H7O, 6H7N, 6IBL, 2Y02, 5F8U, 2YCZ, 3ZPQ, 2Y03, 2Y04, 4AMJ, 4AMI, 2Y01, 2VT4, 2YCY, 4GPO, 2YCX, 6H7M, 5A8E, 3ZPR, 4BVN, 6TKO, 2YCW, 6H7L |
ADRB1 | β1 | 7x48 | 338 | TM7 | F | M | thermostabilising | 2Y00, 6H7J, 6H7O, 6H7N, 6IBL, 2Y02, 5F8U, 2YCZ, 3ZPQ, 2Y03, 2Y04, 4AMJ, 4AMI, 2Y01, 2VT4, 2YCY, 4GPO, 2YCX, 6H7M, 5A8E, 3ZPR, 4BVN, 6TKO, 2YCW, 6H7L |
ADRB1 | β1 | 8x59 | 358 | H8 | C | A | palmitoylation-site | 2Y00, 6H7J, 6H7O, 6H7N, 6IBL, 2Y02, 5F8U, 2YCZ, 3ZPQ, 2Y03, 2Y04, 4AMJ, 4AMI, 2Y01, 2VT4, 2YCY, 4GPO, 2YCX, 6H7M, 5A8E, 3ZPR, 4BVN, 2YCW, 6H7L |
ADRB1 | β1 | 5x58 | 227 | TM5 | Y | A | thermostabilising | 2Y00, 4BVN, 4AMI, 2Y01, 2VT4, 2YCY, 2YCW, 2Y03, 2Y02, 2YCX, 4GPO, 3ZPR, 5F8U, 2YCZ, 3ZPQ, 5A8E, 2Y04, 4AMJ |
ADRB1 | β1 | 6x27 | 282 | TM6 | A | L | thermostabilising | 2Y00, 4BVN, 4AMI, 2Y01, 2VT4, 2YCY, 2YCW, 2Y03, 2Y02, 2YCX, 4GPO, 3ZPR, 5F8U, 2YCZ, 3ZPQ, 5A8E, 2Y04, 4AMJ |
ADRB1 | β1 | 3x40 | 129 | TM3 | I | V | thermostabilising | 4BVN, 5A8E |
ADRB1 | β1 | 3x41 | 130 | TM3 | E | W | thermostabilising | 5A8E |
ADRB1 | β1 | 7x53 | 343 | TM7 | Y | L | thermostabilising | 4BVN, 5A8E |
ADRB1 | β1 | 7x31 | 322 | TM7 | D | K | thermostabilising | 4BVN |
ADRB2 | β2 | 16 | N-term | G | R | other-effect | 3NY8, 3KJ6, 5D6L, 3NY9, 3D4S, 5X7D, 5D5B, 5D5A, 3P0G, 2RH1, 2R4R, 3NYA | |
ADRB2 | β2 | 1x26 | 27 | TM1 | E | Q | other-effect | 3NY8, 3KJ6, 5D6L, 3NY9, 3D4S, 5X7D, 5D5B, 5D5A, 3P0G, 2RH1, 2R4R, 3PDS, 2R4S, 3NYA |
ADRB2 | β2 | 187 | ECL2 | N | E | glycosylation-site | 3NY8, 6E67, 7DHR, 5X7D, 3P0G, 4GBR, 6MXT, 7XKA, 6OBA, 8W1V, 3NYA, 3KJ6, 5D6L, 3NY9, 8JJL, 6PS0, 6PS2, 4QKX, 6N48, 7DHI, 6PS6, 6PS1, 9CHU, 6PRZ, 4LDE, 9CHV, 3SN6, 4LDL, 6PS3, 5JQH, 3D4S, 6PS4, 9CHX, 5D5B, 5D5A, 2RH1, 3PDS, 6PS5, 4LDO, 7XK9 | |
ADRB2 | β2 | 2x66 | 96 | TM2 | M | T | receptor-expression | 4LDE, 4GBR, 4QKX, 4LDL, 3SN6, 5JQH, 4LDO |
ADRB2 | β2 | 23x49 | 98 | ECL1 | M | T | receptor-expression | 4LDE, 4GBR, 4QKX, 4LDL, 3SN6, 5JQH, 4LDO |
ADRB2 | β2 | 6x27 | 265 | TM6 | C | A | other-effect | 4LDE, 4QKX, 4LDL, 5JQH, 4LDO |
ADRB2 | β2 | 3x41 | 122 | TM3 | E | W | thermostabilising, receptor-expression | 3D4S, 3NY8, 3NY9, 3NYA |
ADRB2 | β2 | 2x63 | 93 | TM2 | H | C | thermostabilising, receptor-ligand-bond | 4QKX, 3PDS |
APJ | apelin | 3x40 | 117 | TM3 | V | A | thermostabilising | 5VBL |
APJ | apelin | 177 | ECL2 | T | N | glycosylation-site | 5VBL | |
APJ | apelin | 6x48 | 261 | TM6 | W | K | thermostabilising | 5VBL |
APJ | apelin | 8x59 | 325 | H8 | C | L | palmitoylation-site | 5VBL |
APJ | apelin | 8x60 | 326 | H8 | C | M | palmitoylation-site | 5VBL |
C5AR1 | C5a1 | 2x53 | 85 | TM2 | S | A | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 2x59 | 91 | TM2 | I | A | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 34x51 | 142 | ICL2 | I | A | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 34x55 | 146 | ICL2 | N | R | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 4x45 | 156 | TM4 | A | L | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 4x62 | 172 | TM4 | F | A | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 5x68 | 232 | TM5 | R | A | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 234 | ICL3 | A | E | palmitoylation-site | 5O9H | |
C5AR1 | C5a1 | 8x54 | 311 | H8 | L | E | palmitoylation-site | 5O9H |
C5AR1 | C5a1 | 317 | C-term | S | E | palmitoylation-site | 5O9H | |
C5AR1 | C5a1 | 321 | C-term | N | E | palmitoylation-site | 5O9H | |
CCR5 | CCR5 | 4x61 | 163 | TM4 | G | N | thermostabilising | 7F1Q, 7F1R, 4MBS, 6AKX, 6AKY, 5UIW, 7F1S, 7F1T |
CCR5 | CCR5 | 1x60 | 58 | TM1 | C | Y | thermostabilising | 4MBS, 5UIW, 6AKX, 6AKY, 7F1T |
CCR5 | CCR5 | 6x33 | 233 | TM6 | A | D | thermostabilising, receptor-salt-bridge | 4MBS, 5UIW, 6AKX, 6AKY, 7F1T |
CCR5 | CCR5 | 8x49 | 303 | H8 | K | E | thermostabilising | 4MBS, 5UIW, 6AKX, 6AKY, 7F1T |
CCR9 | CCR9 | 34 | N-term | T | E | glycosylation-site | 5LWE | |
CCR9 | CCR9 | 12x48 | 77 | ICL1 | T | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 12x50 | 79 | ICL1 | V | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 2x38 | 82 | TM2 | M | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 3x47 | 141 | TM3 | S | C | thermostabilising | 5LWE |
CCR9 | CCR9 | 5x41 | 216 | TM5 | T | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 6x36 | 255 | TM6 | V | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 7x29 | 294 | TM7 | N | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 7x39 | 304 | TM7 | T | A | thermostabilising | 5LWE |
CCR9 | CCR9 | 8x63 | 337 | H8 | C | A | palmitoylation-site | 5LWE |
CNR1 | CB1 | 3x46 | 210 | TM3 | T | A | thermostabilising | 5XR8, 5TGZ, 5XRA, 5U09 |
CNR1 | CB1 | 5x37 | 273 | TM5 | E | K | thermostabilising, receptor-expression | 5XR8, 5TGZ, 5XRA |
CNR1 | CB1 | 5x47 | 283 | TM5 | T | V | receptor-expression | 5XR8, 5TGZ, 5XRA |
CNR1 | CB1 | 6x32 | 340 | TM6 | R | E | thermostabilising, receptor-expression | 5XR8, 5TGZ, 5XRA |
CRFR1 | CRF1 | 1x36 | 120 | TM1 | V | A | thermostabilising | 4Z9G, 4K5Y, 8GTI, 8GTG, 8GTM |
CRFR1 | CRF1 | 1x60 | 144 | TM1 | L | A | thermostabilising | 4Z9G, 4K5Y, 8GTI, 8GTG, 8GTM |
CRFR1 | CRF1 | 2x44 | 156 | TM2 | W | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 2x48 | 160 | TM2 | S | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 4x43 | 228 | TM4 | K | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 45x52 | 260 | ECL2 | F | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 5x48 | 277 | TM5 | I | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 6x30 | 309 | TM6 | Y | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 6x51 | 330 | TM6 | F | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 7x38 | 349 | TM7 | S | A | thermostabilising | 4Z9G, 4K5Y |
CRFR1 | CRF1 | 7x53 | 363 | TM7 | Y | A | thermostabilising | 4Z9G, 4K5Y |
CXCR4 | CXCR4 | 3x41 | 125 | TM3 | L | W | thermostabilising | 3OE9, 3OE8, 3OE6, 3OE0, 3ODU, 4RWS |
CXCR4 | CXCR4 | 6x36 | 240 | TM6 | T | P | thermostabilising | 3OE9, 4RWS, 3OE0 |
CXCR4 | CXCR4 | 45x51 | 187 | ECL2 | D | C | thermostabilising, receptor-ligand-bond | 4RWS |
DRD2 | D2 | 3x40 | 122 | TM3 | I | A | thermostabilising | 6CM4 |
DRD2 | D2 | 6x37 | 375 | TM6 | L | A | thermostabilising | 6CM4 |
DRD2 | D2 | 6x41 | 379 | TM6 | L | A | thermostabilising | 6CM4 |
DRD3 | D3 | 3x41 | 119 | TM3 | L | W | thermostabilising | 9F34, 9F33, 3PBL |
EDNRB | ETB | 1x55 | 124 | TM1 | R | Y | thermostabilising | 5XPR, 5X93 |
EDNRB | ETB | 2x56 | 154 | TM2 | D | A | thermostabilising | 5X93 |
EDNRB | ETB | 5x36 | 270 | TM5 | K | A | thermostabilising | 5XPR, 5X93 |
EDNRB | ETB | 6x54 | 342 | TM6 | S | A | thermostabilising | 5XPR, 5X93 |
EDNRB | ETB | 7x48 | 381 | TM7 | I | A | thermostabilising | 5XPR, 5X93 |
EDNRB | ETB | 8x53 | 396 | H8 | C | A | palmitoylation-site | 5XPR, 5X93 |
EDNRB | ETB | 8x57 | 400 | H8 | C | A | palmitoylation-site | 5XPR, 5X93 |
EDNRB | ETB | 405 | C-term | C | A | palmitoylation-site | 5XPR, 5X93 | |
FFAR1 | FFA1 | 2x40 | 42 | TM2 | L | A | thermostabilising | 5TZY, 4PHU, 5TZR, 5KW2 |
FFAR1 | FFA1 | 3x49 | 103 | TM3 | G | A | thermostabilising | 5TZY, 4PHU, 5TZR, 5KW2 |
FFAR1 | FFA1 | 5x58 | 202 | TM5 | Y | F | thermostabilising | 5TZY, 4PHU, 5TZR, 5KW2 |
FFAR1 | FFA1 | 3x34 | 88 | TM3 | F | A | thermostabilising | 5KW2, 4PHU, 5TZR |
GLP1R | GLP-1 | 2x56 | 193 | TM2 | S | C | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 2x59 | 196 | TM2 | I | F | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 3x24 | 225 | TM3 | S | A | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 3x32 | 233 | TM3 | M | C | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 4x48 | 271 | TM4 | S | A | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 5x51 | 317 | TM5 | I | C | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 5x52 | 318 | TM5 | G | I | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 6x30 | 346 | TM6 | K | A | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 6x31 | 347 | TM6 | C | F | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 6x45 | 361 | TM6 | G | C | thermostabilising | 5VEW, 5VEX |
GLP1R | GLP-1 | 207 | ECL1 | T | E | thermostabilising | 5NX2 | |
GLP1R | GLP-1 | 211 | ECL1 | Q | A | thermostabilising | 5NX2 | |
GLP1R | GLP-1 | 215 | ECL1 | D | R | thermostabilising | 5NX2 | |
GLP1R | GLP-1 | 3x31 | 232 | TM3 | L | F | thermostabilising | 5NX2 |
GLP1R | GLP-1 | 260 | ICL2 | L | F | thermostabilising, other-effect | 5NX2 | |
GLP1R | GLP-1 | 295 | ECL2 | G | A | thermostabilising | 5NX2 | |
GLP1R | GLP-1 | 45x52 | 298 | ECL2 | T | A | thermostabilising | 5NX2 |
GLP1R | GLP-1 | 5x63 | 329 | TM5 | C | A | thermostabilising | 5NX2 |
GLP1R | GLP-1 | 6x42 | 358 | TM6 | P | A | thermostabilising | 5NX2 |
GLP1R | GLP-1 | 6x45 | 361 | TM6 | G | A | thermostabilising | 5NX2 |
GLP1R | GLP-1 | 6x47 | 363 | TM6 | H | V | thermostabilising | 5NX2 |
GLP1R | GLP-1 | 7x56 | 405 | TM7 | V | A | thermostabilising | 5NX2 |
GLR | glucagon | 1x48 | 154 | TM1 | G | A | thermostabilising | 5EE7 |
GLR | glucagon | 2x39 | 173 | TM2 | R | A | thermostabilising | 5YQZ, 5EE7 |
GLR | glucagon | 2x48 | 182 | TM2 | A | L | thermostabilising | 5EE7 |
GLR | glucagon | 2x56 | 190 | TM2 | S | A | thermostabilising | 5EE7 |
GLR | glucagon | 2x59 | 193 | TM2 | V | F | thermostabilising | 5EE7 |
GLR | glucagon | 207 | ECL1 | G | E | thermostabilising | 5EE7 | |
GLR | glucagon | 3x24 | 223 | TM3 | G | A | thermostabilising | 5EE7 |
GLR | glucagon | 4x54 | 276 | TM4 | M | A | thermostabilising | 5EE7 |
GLR | glucagon | 6x30 | 344 | TM6 | K | A | thermostabilising | 5EE7 |
GLR | glucagon | 6x48 | 362 | TM6 | E | F | thermostabilising | 5EE7 |
GLR | glucagon | 7x39 | 387 | TM7 | F | A | thermostabilising | 5EE7 |
GRM5 | mGlu5 | 5x42 | 742 | TM5 | T | A | thermostabilising | 8X0F, 7FD8, 6FFI, 4OO9, 8X0H, 7P2L, 8X0E, 6FFH, 5CGD, 8X0D, 8X0C, 8X0B, 8X0G, 7FD9, 5CGC |
GRM5 | mGlu5 | 5x53 | 753 | TM5 | S | A | thermostabilising | 8X0F, 7FD8, 6FFI, 4OO9, 8X0H, 7P2L, 8X0E, 6FFH, 5CGD, 8X0D, 8X0C, 8X0B, 8X0G, 7FD9, 5CGC |
GRM5 | mGlu5 | 1x35 | 579 | TM1 | E | A | thermostabilising | 4OO9, 7P2L, 6FFH, 5CGD, 5CGC, 6FFI |
GRM5 | mGlu5 | 3x48 | 667 | TM3 | N | Y | thermostabilising | 4OO9, 7P2L, 6FFH, 5CGD, 5CGC, 6FFI |
GRM5 | mGlu5 | 3x50 | 669 | TM3 | I | A | thermostabilising | 4OO9, 7P2L, 6FFH, 5CGD, 5CGC, 6FFI |
GRM5 | mGlu5 | 675 | ICL2 | G | M | thermostabilising | 4OO9, 7P2L, 6FFH, 5CGD, 5CGC, 6FFI | |
LPAR1 | LPA1 | 5x37 | 204 | TM5 | D | C | thermostabilising, receptor-disulfide-bridge | 4Z36 |
LPAR1 | LPA1 | 6x59 | 282 | TM6 | V | C | thermostabilising, receptor-disulfide-bridge | 4Z36 |
NPY1R | Y1 | 3x41 | 129 | TM3 | F | W | thermostabilising | 5ZBQ, 5ZBH |
NTR1 | NTS1 | 1x54 | 86 | TM1 | A | L | thermostabilising | 4GRV, 7L0Q, 6ZIN, 6Z8N, 4BV0, 3ZEV, 6Z4Q, 4BWB, 4XES, 7L0P, 6YVR, 8FMZ, 6Z4S, 4XEE, 8FN0, 4BUO, 6Z4V, 7L0S, 6ZA8, 5T04, 6Z66, 7L0R |
NTR1 | NTS1 | 2x40 | 103 | TM2 | H | D | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 2x42 | 105 | TM2 | H | Y | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 3x44 | 161 | TM3 | A | V | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 3x50 | 167 | TM3 | R | L | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 213 | ECL2 | R | L | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV | |
NTR1 | NTS1 | 5x36 | 234 | TM5 | V | L | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 5x54 | 253 | TM5 | I | A | thermostabilising | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 6x32 | 305 | TM6 | H | R | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 7x41 | 358 | TM7 | F | V | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 7x46 | 362 | TM7 | S | A | receptor-expression | 4BWB, 4BUO, 4BV0, 3ZEV |
NTR1 | NTS1 | 215 | ECL2 | G | A | thermostabilising | 4XES, 4XEE, 4GRV, 5T04 | |
NTR1 | NTS1 | 7x43 | 360 | TM7 | V | A | thermostabilising | 4XES, 4XEE, 4GRV, 5T04 |
NTR1 | NTS1 | 1x51 | 83 | TM1 | S | G | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 2x38 | 101 | TM2 | T | R | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 2x551 | 119 | TM2 | L | F | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 2x57 | 121 | TM2 | M | L | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 2x60 | 124 | TM2 | E | D | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 3x26 | 143 | TM3 | R | K | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 3x33 | 150 | TM3 | D | E | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 5x37 | 235 | TM5 | K | R | receptor-expression | 4BWB |
NTR1 | NTS1 | 5x42 | 240 | TM5 | V | L | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 5x61 | 260 | TM5 | I | A | receptor-expression | 4BWB |
NTR1 | NTS1 | 5x63 | 262 | TM5 | N | R | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 5x64 | 263 | TM5 | K | R | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 6x59 | 332 | TM6 | C | V | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 7x25 | 342 | TM7 | F | A | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 7x37 | 354 | TM7 | T | S | receptor-expression | 4BWB, 4BV0 |
NTR1 | NTS1 | 3x49 | 166 | TM3 | E | A | thermostabilising | 4XES, 4GRV |
NTR1 | NTS1 | 2x61 | 125 | TM2 | L | V | receptor-expression | 4BV0 |
NTR1 | NTS1 | 3x55 | 172 | TM3 | C | R | receptor-expression | 4BV0 |
NTR1 | NTS1 | 34x53 | 177 | ICL2 | A | H | receptor-expression | 4BV0 |
NTR1 | NTS1 | 4x65 | 208 | TM4 | M | V | receptor-expression | 4BV0 |
NTR1 | NTS1 | 6x40 | 313 | TM6 | V | M | receptor-expression | 4BV0 |
NTR1 | NTS1 | 7x41 | 358 | TM7 | F | A | receptor-expression | 4GRV, 5T04 |
NTR1 | NTS1 | 6x37 | 310 | TM6 | L | A | thermostabilising | 4GRV |
OPRD | δ | 37 | N-term | P | S | other-effect | 4N6H | |
OPRK | κ | 3x29 | 135 | TM3 | I | L | receptor-expression | 8DZQ, 8DZP, 8DZR, 6VI4, 4DJH, 7YIT, 8DZS, 6B73 |
OPSD | Rhodopsin | 18 | N-term | V | I | other-effect | 2ZIY | |
OPSD | Rhodopsin | 2 | N-term | N | C | thermostabilising, receptor-disulfide-bridge | 6FKC, 4BEY, 5DYS, 6FKA, 6FKB, 6FKD, 6FK7, 2X72, 5EN0, 2J4Y, 6FK8, 4BEZ, 4A4M, 6FK9, 6FK6, 3C9M | |
OPSD | Rhodopsin | 2x56 | 90 | TM2 | G | D | natural-mutation-snp-incl-disease-causing | 4BEZ, 4BEY |
OPSD | Rhodopsin | 282 | ECL3 | D | C | thermostabilising, receptor-disulfide-bridge | 6FKC, 4BEY, 5DYS, 6FKA, 6FKB, 6FKD, 6FK7, 2X72, 5EN0, 2J4Y, 6FK8, 4BEZ, 4A4M, 6FK9, 6FK6, 3C9M | |
OPSD | Rhodopsin | 2x60 | 94 | TM2 | T | I | thermostabilising | 5DYS, 5EN0 |
OPSD | Rhodopsin | 2 | N-term | N | C | thermostabilising, other-effect, receptor-disulfide-bridge | 5DGY, 4ZWJ, 5W0P | |
OPSD | Rhodopsin | 3x28 | 113 | TM3 | E | Q | thermostabilising | 5DGY, 4ZWJ, 5W0P |
OPSD | Rhodopsin | 6x40 | 257 | TM6 | M | Y | thermostabilising | 5DGY, 4ZWJ, 5W0P |
OPSD | Rhodopsin | 282 | ECL3 | N | C | thermostabilising, receptor-disulfide-bridge | 5DGY, 4ZWJ, 5W0P | |
OPSD | Rhodopsin | 6x40 | 257 | TM6 | M | Y | thermostabilising | 4A4M |
OPSD | Rhodopsin | 338 | C-term | S | X | phosphorylation-site | 5W0P | |
OPSD | Rhodopsin | 3x28 | 113 | TM3 | E | Q | thermostabilising | 2X72 |
OX1R | OX1 | 6x56 | 319 | TM6 | V | I | other-effect | 4ZJC, 6V9S, 4ZJ8 |
OX2R | OX2 | 6x39 | 308 | TM6 | I | V | other-effect | 5WQC, 4S0V, 5WS3 |
P2RY1 | P2Y1 | 7x49 | 320 | TM7 | D | N | thermostabilising, receptor-expression | 4XNV, 4XNW |
P2Y12 | P2Y12 | 7x49 | 294 | TM7 | D | N | thermostabilising, receptor-expression | 4NTJ, 4PXZ, 4PY0, 7PP1 |
PAR1 | PAR1 | 250 | ECL2 | N | G | glycosylation-site | 3VW7 | |
PAR1 | PAR1 | 259 | ECL2 | N | S | glycosylation-site | 3VW7 | |
PAR2 | PAR2 | 1x46 | 89 | TM1 | G | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 2x37 | 108 | TM2 | H | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 3x34 | 157 | TM3 | G | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 3x43 | 166 | TM3 | M | L | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 3x51 | 174 | TM3 | Y | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 3x53 | 176 | TM3 | V | E | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 222 | ECL2 | N | Q | glycosylation-site | 5NDZ, 5NJ6, 5NDD | |
PAR2 | PAR2 | 5x64 | 268 | TM5 | M | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 6x38 | 289 | TM6 | I | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PAR2 | PAR2 | 6x42 | 293 | TM6 | L | A | thermostabilising | 5NDZ, 5NJ6, 5NDD |
PTAFR | PAF | 3x51 | 116 | TM3 | F | Y | receptor-expression | 5ZKP, 5ZKQ |
PTAFR | PAF | 169 | ECL2 | N | D | glycosylation-site | 5ZKP, 5ZKQ | |
PTAFR | PAF | 6x34 | 230 | TM6 | A | D | thermostabilising | 5ZKP, 5ZKQ |
PTAFR | PAF | 6x38 | 234 | TM6 | V | A | receptor-expression | 5ZKP, 5ZKQ |
PTAFR | PAF | 7x49 | 289 | TM7 | D | N | receptor-expression | 5ZKP, 5ZKQ |
Q9WTK1 | BLT1 | 2x67 | 83 | TM2 | H | G | thermostabilising | 5X33 |
Q9WTK1 | BLT1 | 3x21 | 88 | TM3 | K | G | thermostabilising | 5X33 |
Q9WTK1 | BLT1 | 5x67 | 212 | TM5 | V | A | thermostabilising | 5X33 |
Q9WTK1 | BLT1 | 309 | C-term | S | A | thermostabilising | 5X33 | |
S1PR1 | S1P1 | 6x30 | 251 | TM6 | S | N | other-effect | 3V2W, 3V2Y |
S1PR1 | S1P1 | 6x31 | 252 | TM6 | L | V | other-effect | 3V2W, 3V2Y |
SMO | SMO | 194 | N-term | E | M | receptor-expression | 5V56 | |
SMO | SMO | 3x40 | 329 | TM3 | V | F | thermostabilising, receptor-expression | 5L7I, 5L7D |
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