Ligand source activities (1 row/activity)
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 1501 | 9561 | 0 | None | - | 1 | Human | 8.4 | pIC50 | None | 8.4 | Functional | Guide to Pharmacology | None | None | None | None | 12401809 | ||||
| 1502 | 9566 | 0 | None | -3 | 2 | Human | 9.0 | pIC50 | None | 9 | Functional | Guide to Pharmacology | None | None | None | None | 12401809 | ||||
| 1496 | 9580 | 0 | None | -15 | 2 | Human | 9.4 | pIC50 | None | 9.4 | Functional | Guide to Pharmacology | None | None | None | None | 12401809 | ||||
| 1495 | 9579 | 0 | None | -2 | 2 | Human | 9.6 | pIC50 | None | 9.6 | Functional | Guide to Pharmacology | None | None | None | None | 12401809 | ||||
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |