Ligand source activities (1 row/activity)





Ligands Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb ID #Vendors Reference
ligand
Fold selectivity
(Potency)
# tested GPCRs
(Potency)
Species p-value
(-log)
Type Activity
Relation
Activity
Value
Assay Type Assay Description Source Mol
weight
Rot
Bonds
H don H acc LogP Smiles DOI
5572 8709 0 None - 1 Rat 7.6 pA2 = 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None None
129631922 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
132274287 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
132451761 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
155817470 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
16132393 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
16133850 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
4448 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
4514 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
91933454 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
CHEMBL525610 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
DB06285 10553 13 None -34 4 Rat 8.2 pIC50 = 8.2 Functional
NoneNone
Drug Central None None None None None
129631922 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
132274287 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
132451761 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
155817470 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
16132393 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
16133850 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
4448 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
4514 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
91933454 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
CHEMBL525610 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
DB06285 10553 13 None -7 4 Human 8.1 pIC50 = 8.1 Functional
NoneNone
Drug Central None None None None None
155817427 10006 0 None -158 3 Rat 5.5 pIC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1788 10006 0 None -158 3 Rat 5.5 pIC50 = 5.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129316189 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817471 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16201228 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4449 10003 0 None -35 3 Rat 6.8 pIC50 = 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1824 8784 0 None - 1 Human 7.0 pIC50 = 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
155817427 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817427 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1788 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1788 10006 0 None -1 3 Human 7.5 pIC50 = 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
129631922 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129631922 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
132274287 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132274287 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
132451761 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132451761 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817470 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817470 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
16132393 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16132393 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
16133850 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16133850 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
4448 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4448 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
4514 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4514 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
91933454 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
91933454 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
CHEMBL525610 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
CHEMBL525610 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
DB06285 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
DB06285 10553 13 None -7 4 Human 7.8 pIC50 = 7.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
3624 10597 0 None -5 2 Rat 8.1 pIC50 = 8.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1815 10598 0 None 25 3 Human 8.4 pIC50 = 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
1815 10598 0 None 25 3 Human 8.4 pIC50 = 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
3624 10597 0 None 5 2 Human 8.8 pIC50 = 8.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817432 10007 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16144017 10007 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1822 10007 0 None -446 3 Rat 5.3 pIC50 None 5.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817428 10008 0 None -6 2 Human 5.7 pIC50 None 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1790 10008 0 None -6 2 Human 5.7 pIC50 None 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817432 10007 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16144017 10007 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1822 10007 0 None -70 3 Human 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817433 10600 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16134968 10600 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1827 10600 0 None -125 3 Rat 6.1 pIC50 None 6.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1825 8777 0 None - 1 Human 6.2 pIC50 None 6.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1820 8279 0 None -10 2 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1807 9878 0 None -5 2 Human 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
129631922 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132274287 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
132451761 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817470 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16132393 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16133850 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4448 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4514 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
91933454 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
CHEMBL525610 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
DB06285 10553 13 None -34 4 Rat 6.3 pIC50 None 6.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817434 10601 0 None -50 2 Rat 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1828 10601 0 None -50 2 Rat 6.5 pIC50 None 6.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1794 8711 0 None 19 3 Human 6.6 pIC50 None 6.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
155817429 10009 0 None -3 2 Human 6.7 pIC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1814 10009 0 None -3 2 Human 6.7 pIC50 None 6.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1801 8782 0 None -3 2 Human 6.8 pIC50 None 6.8 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1819 8280 0 None -3 2 Human 6.9 pIC50 None 6.9 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1821 8783 0 None -1 2 Human 7.0 pIC50 None 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1815 10598 0 None -25 3 Rat 7.0 pIC50 None 7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817433 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
155817433 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16134968 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
16134968 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1827 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11046116
1827 10600 0 None -12 3 Human 7.1 pIC50 None 7.1 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1800 8781 0 None -3 2 Human 7.2 pIC50 None 7.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1820 8279 0 None 10 2 Human 7.3 pIC50 None 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1799 8780 0 None -1 2 Human 7.3 pIC50 None 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1808 10644 0 None 2 2 Human 7.4 pIC50 None 7.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9360953
1809 10643 0 None 1 2 Human 7.5 pIC50 None 7.5 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1798 8779 0 None -1 2 Human 7.6 pIC50 None 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
1798 8779 0 None -1 2 Human 7.6 pIC50 None 7.6 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 8702701
1797 8785 0 None 1 2 Human 7.7 pIC50 None 7.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 9360953
155817434 10601 0 None 50 2 Human 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
1828 10601 0 None 50 2 Human 8.2 pIC50 None 8.2 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
129316189 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
129316189 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
129316189 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
155817471 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
155817471 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
155817471 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
16201228 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
16201228 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
16201228 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681
4449 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10537121
4449 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 10854439
4449 10003 0 None 15 3 Human 8.4 pIC50 None 8.4 Functional
UnclassifiedUnclassified
Guide to Pharmacology None None None None 11602681




Ligands Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb ID #Vendors Reference
ligand
Fold selectivity
(Affinity)
# tested GPCRs
(Affinity)
Species p-value
(-log)
Type Activity
Relation
Activity
Value
Assay Type Assay Description Source Mol
weight
Rot
Bonds
H don H acc LogP Smiles DOI