CXCR2

GPCR CLASS (FAMILY)

Class A (Rhodopsin)

PDB CODE

SPECIES

Homo sapiens

RESOLUTION

3.2 Å

PREFERRED CHAIN

A

REFERENCE

PUBLICATION DATE

Sept. 2, 2020

3D VIEW

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LIGAND INTERACTIONS

LIGANDS

4-[[3,4-Dioxo-2-[[(1R)-1-(4-propan-2-ylfuran-2-yl)propyl]amino]cyclobuten-1-yl]amino]-3-hydroxy-N,N-dimethylpyridine-2-carboxamide - Allosteric antagonist pubchem

ENDOGENOUS LIGANDS

CXCL5, CXCL3, CXCL6, CXCL2, CXCL1, CXCL8, CXCL7