SRIF-28
SMILES | None |
InChIKey | GGYTXJNZMFRSLX-DFTNLTQTSA-N |
Sequence | SANSNPAMAPRERKAGCKNFFWKTFTSC |
Chemical properties
Hydrogen bond acceptors | None |
Hydrogen bond donors | None |
Rotatable bonds | None |
Molecular weight (Da) |
Drug properties
Molecular type | Peptide |
Physiological/Surrogate | Endogenous |
Approved drug | No |
Database connections
Sankey plot
Compound is not listed as a drug.
Bioactivities
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
SST1 | SSR1 | Human | Somatostatin | A | pKi | 8.6 | 9.0 | 9.4 | Guide to Pharmacology |
SST2 | SSR2 | Human | Somatostatin | A | pKi | 8.4 | 9.3 | 10.2 | Guide to Pharmacology |
SST3 | SSR3 | Human | Somatostatin | A | pKi | 8.1 | 9.0 | 9.9 | Guide to Pharmacology |
SST4 | SSR4 | Human | Somatostatin | A | pKi | 8.1 | 8.65 | 9.2 | Guide to Pharmacology |
SST5 | SSR5 | Human | Somatostatin | A | pKi | 9.2 | 9.75 | 10.3 | Guide to Pharmacology |
SST5 | SSR5 | Rat | Somatostatin | A | pKi | 9.0 | 9.0 | 9.0 | Guide to Pharmacology |
SST2 | SSR2 | Rat | Somatostatin | A | pKi | 8.8 | 8.8 | 8.8 | Guide to Pharmacology |
SST5 | SSR5 | Mouse | Somatostatin | A | pKi | 9.8 | 9.85 | 9.9 | Guide to Pharmacology |
SST3 | SSR3 | Rat | Somatostatin | A | pKi | 9.1 | 9.1 | 9.1 | Guide to Pharmacology |
Receptor | Activity | Source | |||||||
---|---|---|---|---|---|---|---|---|---|
GTP | Uniprot | Species | Family | Class | Type | Min | Avg | Max | Database |
SST3 | SSR3 | Mouse | Somatostatin | A | pIC50 | 10.2 | 10.2 | 10.2 | Guide to Pharmacology |
SST2 | SSR2 | Mouse | Somatostatin | A | pIC50 | 9.0 | 9.25 | 9.5 | Guide to Pharmacology |
SST2 | SSR2 | Human | Somatostatin | A | pEC50 | 8.64 | 8.64 | 8.64 | ChEMBL |
MRGPRX2 | MRGX2 | Human | A orphans | A | pEC50 | 5.38 | 5.38 | 5.38 | Guide to Pharmacology |