GPCRdb

CHEMBL415165

Agent/drug
Bioactivity

CHEMBL415165

No image available

SMILES	None
InChIKey	BUVGQEXSQXRZQG-LBQSHGEUSA-N

Chemical Properties

Hydrogen bond acceptors	None
Hydrogen bond donors	None
Rotatable bonds	None
Molecular weight (Da)

Database connections

ChEMBL_compound_ids GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

MC₁	MSHR	Human	Melanocortin	A	pKi	10.00	10.00	10.00	ChEMBL
MC₃	MC3R	Human	Melanocortin	A	pKi	9.64	9.64	9.64	ChEMBL
MC₄	MC4R	Rat	Melanocortin	A	pKi	10.05	10.05	10.05	ChEMBL
MC₄	MC4R	Human	Melanocortin	A	pKi	9.51	9.51	9.51	ChEMBL
MC₅	MC5R	Human	Melanocortin	A	pKi	9.77	9.77	9.77	ChEMBL

Showing 1 to 5 of 5 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

MC₄	MC4R	Human	Melanocortin	A	pEC50	9.44	9.58	9.72	ChEMBL

Showing 1 to 1 of 1 entry

CHEMBL415165

No image available

Drug properties

Molecular type	Protein
Physiological/Surrogate	Surrogate
Approved drug	No

Distribution across phases (no. indications)

Phase I 0

Phase II 0

Phase III 0

Phase IV

Database connections

ChEMBL_compound_ids GPCRdb

Compound is not listed as a drug.