GPCRdb

methimepip

Agent/drug
Bioactivity

methimepip

SMILES	CN1CCC(Cc2cnc[nH]2)CC1
InChIKey	KIAVPENCSGKVQP-UHFFFAOYSA-N

Chemical Properties

Hydrogen bond acceptors	2
Hydrogen bond donors	1
Rotatable bonds	2
Molecular weight (Da)	179.1

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

H₃	HRH3	Human	Histamine	A	pKi	9.00	9.00	9.00	Guide to Pharmacology
H₃	HRH3	Human	Histamine	A	pKi	9.00	9.00	9.00	ChEMBL
H₄	HRH4	Human	Histamine	A	pKi	5.70	5.70	5.70	Guide to Pharmacology
H₄	HRH4	Human	Histamine	A	pKi	5.70	5.70	5.70	ChEMBL

Showing 1 to 4 of 4 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

H₃	HRH3	Human	Histamine	A	pEC50	9.50	9.50	9.50	ChEMBL
H₄	HRH4	Human	Histamine	A	pEC50	5.30	5.30	5.30	ChEMBL

Showing 1 to 2 of 2 entries

methimepip

Drug properties

Molecular type	Small molecule
Physiological/Surrogate	Surrogate
Approved drug	No

Distribution across phases (no. indications)

Phase I 0

Phase II 0

Phase III 0

Phase IV

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Compound is not listed as a drug.