GPCRdb

milameline

Agent/drug
Bioactivity

milameline

SMILES	CO/N=C/C1=CCCN(C)C1
InChIKey	YMMXHEYLRHNXAB-RMKNXTFCSA-N

Chemical Properties

Hydrogen bond acceptors	3
Hydrogen bond donors	0
Rotatable bonds	2
Molecular weight (Da)	154.1

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

M₁	ACM1	Human	Acetylcholine (muscarinic)	A	pKi	5.25	5.25	5.25	ChEMBL
M₁	ACM1	Human	Acetylcholine (muscarinic)	A	pKi	4.80	4.80	4.80	Guide to Pharmacology
M₂	ACM2	Human	Acetylcholine (muscarinic)	A	pKi	6.00	6.00	6.00	ChEMBL
M₃	ACM3	Human	Acetylcholine (muscarinic)	A	pKi	5.10	5.10	5.10	Guide to Pharmacology
M₄	ACM4	Human	Acetylcholine (muscarinic)	A	pKi	5.50	5.50	5.50	Guide to Pharmacology
M₅	ACM5	Human	Acetylcholine (muscarinic)	A	pKi	5.40	5.40	5.40	Guide to Pharmacology
M₅	ACM5	Human	Acetylcholine (muscarinic)	A	pKi	5.50	5.50	5.50	ChEMBL

Showing 1 to 7 of 7 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

M₁	ACM1	Human	Acetylcholine (muscarinic)	A	pEC50	7.68	7.68	7.68	ChEMBL

Showing 1 to 1 of 1 entry

milameline

Drug properties

Molecular type	Small molecule
Physiological/Surrogate	Surrogate
Approved drug	No

Distribution across phases (no. indications)

Phase I 0

Phase II 0

Phase III 0

Phase IV

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Compound is not listed as a drug.