GPCRdb

naltriben

Agent/drug
Bioactivity

naltriben

SMILES	Oc1ccc2c3c1O[C@H]1c4oc5ccccc5c4C[C@@]4(O)[C@@H](C2)N(CC2CC2)CC[C@]314
InChIKey	ZHVWWEYETMPAMX-IFKAHUTRSA-N

Chemical Properties

Hydrogen bond acceptors	5
Hydrogen bond donors	2
Rotatable bonds	2
Molecular weight (Da)	415.2

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids Guide To Pharmacology GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

δ	OPRD	Human	Opioid	A	pKi	10.00	10.00	10.00	Guide to Pharmacology
δ	OPRD	Rat	Opioid	A	pKi	10.00	10.00	10.00	Guide to Pharmacology
δ	OPRD	Mouse	Opioid	A	pKi	10.90	10.90	10.90	Guide to Pharmacology
δ	OPRD	Human	Opioid	A	pKi	10.89	10.89	10.89	ChEMBL
κ	OPRK	Human	Opioid	A	pKi	8.40	8.40	8.40	Guide to Pharmacology
κ	OPRK	Guinea pig	Opioid	A	pKi	6.82	6.82	6.82	ChEMBL
μ	OPRM	Human	Opioid	A	pKi	7.90	7.90	7.90	Guide to Pharmacology

Showing 1 to 7 of 7 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

κ	OPRK	Human	Opioid	A	pIC50	6.16	6.16	6.16	ChEMBL

Showing 1 to 1 of 1 entry

naltriben

Drug properties

Molecular type	Small molecule
Physiological/Surrogate	Surrogate
Approved drug	No

Distribution across phases (no. indications)

Phase I 0

Phase II 0

Phase III 0

Phase IV 0

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids Guide To Pharmacology GPCRdb

Compound is not listed as a drug.