GPCRdb

SB 207710

Agent/drug
Bioactivity

SB 207710

SMILES	CCCCN1CCC(COC(=O)c2cc(I)c(N)c3c2OCCO3)CC1
InChIKey	FCKKCDRMGKXQDK-UHFFFAOYSA-N

Chemical Properties

Hydrogen bond acceptors	6
Hydrogen bond donors	1
Rotatable bonds	6
Molecular weight (Da)	474.1

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

5-HT₄	5HT4R	Human	5-Hydroxytryptamine	A	pKi	10.10	10.20	10.30	Guide to Pharmacology
5-HT₄	5HT4R	Rat	5-Hydroxytryptamine	A	pKd	9.52	9.52	9.52	ChEMBL
5-HT₄	5HT4R	Human	5-Hydroxytryptamine	A	pKi	8.66	8.66	8.66	ChEMBL
5-HT₇	5HT7R	Human	5-Hydroxytryptamine	A	pKi	5.30	5.40	5.50	Guide to Pharmacology

Showing 1 to 4 of 4 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

5-HT₄	5HT4R	Human	5-Hydroxytryptamine	A	pEC50	7.90	7.90	7.90	ChEMBL

Showing 1 to 1 of 1 entry

SB 207710

Drug properties

Molecular type	Small molecule
Physiological/Surrogate	Surrogate
Approved drug	No

Distribution across phases (no. indications)

Phase I 0

Phase II 0

Phase III 0

Phase IV 0

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Compound is not listed as a drug.