GPCRdb

seglitide

Agent/drug
Bioactivity

seglitide

SMILES	None
InChIKey	NPJIOCBFOAHEDO-AVWFULIKSA-N
Sequence	AYWKVF

Chemical Properties

Hydrogen bond acceptors	None
Hydrogen bond donors	None
Rotatable bonds	None
Molecular weight (Da)

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Bioactivities

Affinity
Potency

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

SST2	SSR2	Human	Somatostatin	A	pKi	8.80	9.55	10.30	Guide to Pharmacology
SST2	SSR2	Rat	Somatostatin	A	pKi	9.30	9.30	9.30	Guide to Pharmacology
SST2	SSR2	Mouse	Somatostatin	A	pKi	7.10	8.50	9.90	Guide to Pharmacology
SST2	SSR2	Human	Somatostatin	A	pKi	9.52	9.81	10.10	ChEMBL
SST3	SSR3	Human	Somatostatin	A	pKi	6.60	7.25	7.90	Guide to Pharmacology
SST3	SSR3	Rat	Somatostatin	A	pKi	7.40	7.40	7.40	Guide to Pharmacology
SST3	SSR3	Human	Somatostatin	A	pKi	7.50	7.50	7.50	ChEMBL
SST4	SSR4	Human	Somatostatin	A	pKi	5.50	5.50	5.50	ChEMBL
SST5	SSR5	Human	Somatostatin	A	pKi	6.60	8.40	10.20	Guide to Pharmacology
SST5	SSR5	Rat	Somatostatin	A	pKi	7.10	7.10	7.10	Guide to Pharmacology
SST5	SSR5	Mouse	Somatostatin	A	pKi	6.70	7.60	8.50	Guide to Pharmacology
SST5	SSR5	Human	Somatostatin	A	pKi	7.90	7.90	7.90	ChEMBL

Showing 1 to 12 of 12 entries

Search:

Receptor					Activity				Source

Protein	Gene	Species	Family	Class	Type	Min	Avg	Max	Database

SST2	SSR2	Human	Somatostatin	A	pIC50	8.80	8.80	8.80	ChEMBL
SST3	SSR3	Mouse	Somatostatin	A	pIC50	7.90	7.90	7.90	Guide to Pharmacology
SST3	SSR3	Human	Somatostatin	A	pIC50	6.98	6.98	6.98	ChEMBL
SST5	SSR5	Human	Somatostatin	A	pIC50	7.09	7.09	7.09	ChEMBL

Showing 1 to 4 of 4 entries

seglitide

Drug properties

Molecular type	Peptide
Physiological/Surrogate	Surrogate
Approved drug	No

Distribution across phases (no. indications)

Phase I 0

Phase II 0

Phase III 0

Phase IV 0

Database connections

PubChem Guide To Pharmacology ChEMBL_compound_ids GPCRdb

Compound is not listed as a drug.