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Ligand source activities (1 row/activity)

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	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

Ligands				Receptor	Activity									Chemical information
Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

α-methyl-5-HT	364	None	24	Human	Binding	pKi	None	-	6.70	-25	19	Unclassified	Guide to Pharmacology	190.1	2	3	2	1.76	CC(N)Cc1c[nH]c2ccc(O)cc12	https://pubmed.ncbi.nlm.nih.gov/8380639
α-methyl-5-HT	364	3H-5HT	24	Human	Binding	pKi	=	184.00	6.74	-25	19	-	PDSP KiDatabase	190.1	2	3	2	1.76	CC(N)Cc1c[nH]c2ccc(O)cc12	-
α-methyl-5-HT	364	3H-5HT	24	Human	Binding	pKi	=	181.97	6.74	-25	19	-	PDSP KiDatabase	190.1	2	3	2	1.76	CC(N)Cc1c[nH]c2ccc(O)cc12	-
1-naphthylpiperazine	35	3H-5HT	37	Human	Binding	pKi	=	53.70	7.27	-21	21	-	PDSP KiDatabase	212.1	1	1	2	2.25	c1ccc2c(N3CCNCC3)cccc2c1	-
1-naphthylpiperazine	35	3H-5HT	37	Human	Binding	pKi	=	54.00	7.27	-21	21	-	PDSP KiDatabase	212.1	1	1	2	2.25	c1ccc2c(N3CCNCC3)cccc2c1	-
1-naphthylpiperazine	35	None	37	Human	Binding	pKi	None	-	7.30	-21	21	Unclassified	Guide to Pharmacology	212.1	1	1	2	2.25	c1ccc2c(N3CCNCC3)cccc2c1	https://pubmed.ncbi.nlm.nih.gov/8380639
1-naphthylpiperazine	35	None	37	Human	Binding	pKi	None	-	7.30	-21	21	Unclassified	Guide to Pharmacology	212.1	1	1	2	2.25	c1ccc2c(N3CCNCC3)cccc2c1	https://pubmed.ncbi.nlm.nih.gov/9225282
2-methyl-5-HT	81	None	43	Human	Binding	pKi	None	-	6.40	-4	21	Unclassified	Guide to Pharmacology	190.1	2	3	2	1.68	Cc1[nH]c2ccc(O)cc2c1CCN	https://pubmed.ncbi.nlm.nih.gov/8380639
2-methyl-5-HT	81	3H-5HT	43	Human	Binding	pKi	=	413.00	6.38	-4	21	-	PDSP KiDatabase	190.1	2	3	2	1.68	Cc1[nH]c2ccc(O)cc2c1CCN	-
2-methyl-5-HT	81	3H-5HT	43	Human	Binding	pKi	=	416.86	6.38	-4	21	-	PDSP KiDatabase	190.1	2	3	2	1.68	Cc1[nH]c2ccc(O)cc2c1CCN	-
5-BODMT	129	None	0	Human	Binding	pKi	=	-	8.44	66	2	Unclassified	Guide to Pharmacology	272.2	7	1	2	3.18	CCCC(=O)Cc1ccc2[nH]cc(CCN(C)C)c2c1	https://pubmed.ncbi.nlm.nih.gov/21422162
5-CT	134	None	25	Human	Binding	pKi	None	-	6.10	-8317	39	Unclassified	Guide to Pharmacology	203.1	3	3	2	0.77	NCCc1c[nH]c2ccc(C(N)=O)cc12	https://pubmed.ncbi.nlm.nih.gov/8380639
5-CT	134	None	25	Human	Binding	pKi	None	-	6.10	-8317	39	Unclassified	Guide to Pharmacology	203.1	3	3	2	0.77	NCCc1c[nH]c2ccc(C(N)=O)cc12	https://pubmed.ncbi.nlm.nih.gov/9225282
5-CT	134	3H-5HT	25	Human	Binding	pKi	=	724.43	6.14	-8317	39	-	PDSP KiDatabase	203.1	3	3	2	0.77	NCCc1c[nH]c2ccc(C(N)=O)cc12	-
5-CT	134	3H-5HT	25	Human	Binding	pKi	=	717.00	6.14	-8317	39	-	PDSP KiDatabase	203.1	3	3	2	0.77	NCCc1c[nH]c2ccc(C(N)=O)cc12	-
5-CT	134	125I-LSD	25	Mouse	Binding	pKi	=	3162.27	5.50	-34673	39	-	PDSP KiDatabase	203.1	3	3	2	0.77	NCCc1c[nH]c2ccc(C(N)=O)cc12	-
5-CT	134	125I-LSD	25	Rat	Binding	pKi	=	2454.70	5.61	-26915	39	-	PDSP KiDatabase	203.1	3	3	2	0.77	NCCc1c[nH]c2ccc(C(N)=O)cc12	-
5-hydroxytryptamine	139	None	45	Human	Binding	pKi	None	-	7.85	-144	61	Unclassified	Guide to Pharmacology	176.1	2	3	2	1.38	NCCc1c[nH]c2ccc(O)cc12	https://pubmed.ncbi.nlm.nih.gov/15900510
5-hydroxytryptamine	139	None	45	Human	Binding	pKi	None	-	7.85	-144	61	Unclassified	Guide to Pharmacology	176.1	2	3	2	1.38	NCCc1c[nH]c2ccc(O)cc12	https://pubmed.ncbi.nlm.nih.gov/8380639
5-hydroxytryptamine	139	None	45	Human	Binding	pKi	None	-	7.85	-144	61	Unclassified	Guide to Pharmacology	176.1	2	3	2	1.38	NCCc1c[nH]c2ccc(O)cc12	https://pubmed.ncbi.nlm.nih.gov/9225282

Showing 1 to 20 of 293 entries

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

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Ligand source activities (1 row/activity)