Ligand source activities (1 row/activity)
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 125957 | 126938 | 8 | None | 1 | 2 | Rat | 7.2 | pKi | = | 7.2 | Binding | ChEMBL | 256 | 0 | 1 | 2 | 2.4 | FC(F)(F)c1ccc2c(c1)N1CCNCC1CC2 | 10.1016/S0960-894X(97)00074-7 | ||
| CHEMBL351530 | 126938 | 8 | None | 1 | 2 | Rat | 7.2 | pKi | = | 7.2 | Binding | ChEMBL | 256 | 0 | 1 | 2 | 2.4 | FC(F)(F)c1ccc2c(c1)N1CCNCC1CC2 | 10.1016/S0960-894X(97)00074-7 | ||