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Ligand source activities (1 row/activity)

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	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

Ligands				Receptor	Activity									Chemical information
Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

[p-aminoPhe6]ang II	2996	None	0	Rat	Binding	pKd	=	-	9.26	-	1	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/2194459
ANGIOTENSIN	212871	None	0	Human	Binding	IC50	=	0.13	9.89	-	1	Binding affinity to human angiotensin AT2 receptor by radioligand displacement assay	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1016/j.bmc.2013.03.016
angiotensin A	418	None	0	Human	Binding	pKi	=	-	8.64	-1	3	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/21464395
angiotensin II	419	None	38	Human	Binding	pKd	=	-	10.20	1	5	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/2775266
angiotensin II	419	None	38	Human	Binding	pKd	=	-	10.20	1	5	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/7850406
angiotensin II	419	None	38	Human	Binding	pKd	=	10.20	7.99	1	5	None	Drug Central	-	-	-	-	-	-	-
angiotensin II	419	None	38	Human	Binding	IC50	=	0.62	9.21	1	5	Displacement of [125-I]-[Sar1, Ile8] from recombinant human AT2R transfected in human HEK293 cells incubated for 2 hrs by liquid scintillation counter analysis	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1016/j.bmcl.2021.128086
angiotensin II	419	None	38	Human	Binding	IC50	=	0.08	10.10	1	5	Displacement of [125I]CGP 42112A from human recombinant AT2 receptor expressed in HEK293 cells measured after 4 hrs by scintillation counting method	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1016/j.bmc.2016.11.014
angiotensin II	419	None	38	Human	Binding	Ki	=	0.20	9.70	1	5	Binding affinity to type-2 angiotensin-2 receptor (unknown origin)	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1016/j.bmcl.2015.10.084
angiotensin II	419	None	38	Human	Binding	Ki	=	0.30	9.52	1	5	Displacement of [125I]Ang2 from AT2 receptor in pig uterus myometrial membrane	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm0613469
angiotensin II	419	None	38	Human	Binding	Ki	=	0.60	9.22	1	5	Displacement of [125I]Ang2 from AT2 receptor in pig uterus myometrium	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm051222g
angiotensin II	419	None	38	Human	Binding	Ki	=	0.20	9.70	1	5	Binding affinity for angiotensin II receptor, type 2 in pig uterus myometrium using [125I]-Ang II as radioligand, in pH 7.4 Tris-HCl buffer for 1.5 hr at 25 degree C	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm050280z
angiotensin II	419	None	38	Human	Binding	Ki	=	0.23	9.64	1	5	Displacement of [125I]-Ang II from angiotensin II receptor type 2 in pig uterus myometrium	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm0491492
angiotensin II	419	None	38	Human	Binding	Ki	=	1.20	8.92	1	5	Displacement of [125I]-Ang II from pig uterus myometrium angiotensin II type 2 (AT2) receptor	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm049651m
angiotensin II	419	None	38	Human	Binding	Ki	=	0.23	9.64	1	5	Binding affinity for Angiotensin II receptor type 2 using [125I]- Ang II in pig uterus myometrium	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm030921v
angiotensin II	419	None	38	Human	Binding	IC50	=	2.50	8.60	1	5	In vitro binding affinity at angiotensin II (type 2) receptor in rabbit uterus.	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm00065a013
angiotensin III	420	None	0	Human	Binding	pKd	=	-	10.40	-	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/8242249
angiotensin III	420	None	0	Human	Binding	pKd	=	-	10.40	-	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/2775266
angiotensin III	420	None	0	Human	Binding	IC50	=	1.74	8.76	-	2	In vitro binding affinity at angiotensin II (type 2) receptor in rabbit uterus.	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1021/jm00065a013
ANGIOTENSIN-II	212873	None	5	Human	Binding	Ki	=	0.11	9.96	-	3	Binding affinity to human AT2 receptor by radioligand displacement assay	ChEMBL	-	-	-	-	-	-	https://dx.doi.org/10.1016/j.ejmech.2013.01.044

Showing 1 to 20 of 1,205 entries

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

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Ligand source activities (1 row/activity)