Ligand source activities (1 row/activity)
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 1023 | 1643 | 0 | None | -10000 | 5 | Human | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | None | None | None | None | 16025565 | ||||
| 3935 | 1588 | 0 | None | 50 | 2 | Human | 8.1 | pEC50 | = | 8.1 | Functional | Guide to Pharmacology | None | None | None | None | 15623572 | ||||
| 1048 | 4022 | 0 | None | -11 | 4 | Human | 8.5 | pEC50 | = | 8.5 | Functional | Guide to Pharmacology | None | None | None | None | 11285256 | ||||
| 1046 | 1910 | 0 | None | - | 1 | Human | 5.0 | pEC50 | None | 5 | Functional | Guide to Pharmacology | None | None | None | None | 11602630 | ||||
| 155817387 | 1910 | 0 | None | - | 1 | Human | 5.0 | pEC50 | None | 5 | Functional | Guide to Pharmacology | None | None | None | None | 11602630 | ||||
| 16131967 | 1910 | 0 | None | - | 1 | Human | 5.0 | pEC50 | None | 5 | Functional | Guide to Pharmacology | None | None | None | None | 11602630 | ||||
| 1044 | 421 | 0 | None | 1 | 3 | Human | 6.0 | pEC50 | None | 6 | Functional | Guide to Pharmacology | None | None | None | None | 15187149 | ||||
| 1047 | 1921 | 13 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| 16131438 | 1921 | 13 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| 56947109 | 1921 | 13 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| CHEMBL4447799 | 1921 | 13 | None | 3 | 4 | Human | 9.0 | pEC50 | None | 9.0 | Functional | Guide to Pharmacology | None | None | None | None | 15465011 | ||||
| 1040 | 4031 | 0 | None | -4 | 2 | Human | 6.0 | pIC50 | None | 6 | Functional | Guide to Pharmacology | None | None | None | None | 16476585 | ||||
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |