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Ligand source activities (1 row/activity)

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	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

Ligands				Receptor	Activity									Chemical information
Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

1-(benzo[d]thiazol-2-yl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine	220110	UNDEFINED	0	Human	Binding	pKi	=	10000.00	5.00	-1	3	-	PDSP KiDatabase	383.2	6	1	6	4.78	CCOc1cc(NC2CCN(c3nc4ccccc4s3)CC2)ccc1OC	-
1-(benzo[d]thiazol-2-ylmethyl)-N-(3-ethoxy-4-methoxyphenyl)piperidin-4-amine	220111	UNDEFINED	0	Human	Binding	pKi	=	10000.00	5.00	-1	3	-	PDSP KiDatabase	397.2	7	1	6	4.78	CCOc1cc(NC2CCN(Cc3nc4ccccc4s3)CC2)ccc1OC	-
2-(4-((4-(benzo[d]oxazol-2-ylamino)piperidin-1-yl)methyl)-2-ethoxy-5-fluorophenoxy)ethanol	220122	UNDEFINED	0	Human	Binding	pKi	=	10000.00	5.00	-1	3	-	PDSP KiDatabase	429.2	9	2	7	3.81	CCOc1cc(CN2CCC(Nc3nc4ccccc4o3)CC2)c(F)cc1OCCO	-
[D-Tyr⁸]CYN 154806	1506	None	0	Human	Binding	pKi	=	-	6.45	-112	6	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/10818261
[L-Tyr⁸]CYN 154806	2375	None	0	Human	Binding	pKi	=	-	6.50	-56	6	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/10818261
ACQ090	266	None	0	Human	Binding	pKi	=	-	7.90	-	1	Unclassified	Guide to Pharmacology	526.3	7	0	5	4.63	COc1ccc(CC(C)CN2C[C@@H](C(=O)N3CCN(c4ccc(F)c(F)c4)CC3)[C@H]3CCCC[C@H]3C2)cn1	-
astemizole	505	UNDEFINED	55	Human	Binding	pKi	=	10000.00	5.00	-5754	48	-	PDSP KiDatabase	458.2	8	1	5	5.35	COc1ccc(CCN2CCC(Nc3nc4ccccc4n3Cc3ccc(F)cc3)CC2)cc1	-
BIM 23023	637	None	0	Human	Binding	pKi	=	-	8.10	-19	8	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/7988476
BIM 23023	637	None	0	Rat	Binding	pKi	=	-	7.00	-251	8	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/9600011
BIM 23030	639	None	0	Human	Binding	pKi	=	-	7.50	-1	5	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/9650799
BIM 23030	639	None	0	Human	Binding	pKi	=	-	7.50	-1	5	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/10598788
BIM 23034	640	None	0	Human	Binding	pKi	=	-	8.10	-3	4	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/7988476
BIM 23050	641	None	0	Human	Binding	pKi	=	-	7.80	-10	4	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/7988476
BIM 23052	642	None	0	Human	Binding	pKi	=	-	9.05	2	9	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/8769372
BIM 23052	642	None	0	Human	Binding	pKi	=	-	9.05	2	9	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/9650799
BIM 23052	642	None	0	Human	Binding	pKi	=	-	9.05	2	9	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/10598788
BIM 23052	642	None	0	Rat	Binding	pKi	=	-	8.50	-3	9	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/9600011
BIM 23056	643	None	0	Human	Binding	pKi	=	-	7.05	-4	7	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/9650799
BIM 23056	643	None	0	Human	Binding	pKi	=	-	7.05	-4	7	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/10598788
BIM 23058	644	None	0	Human	Binding	pKi	=	-	8.80	-	2	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/7988476

Showing 1 to 20 of 1,068 entries

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

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Ligand source activities (1 row/activity)