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Ligand source activities (1 row/activity)

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	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

Ligands				Receptor	Activity									Chemical information
Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

CHEMBL1235128	16490	None	4	Rat	Binding	Ki	=	31.00	7.51	-2	7	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	322.1	4	4	9	-1.45	CCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL129903	19496	None	0	Rat	Binding	Ki	=	167.00	6.78	-3	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	323.1	4	5	10	-2.90	NCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL1791423	63282	None	0	Rat	Binding	Ki	=	20.00	7.70	44	3	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	291.1	2	4	9	-1.98	C#CC(O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL2070507	76962	None	0	Rat	Binding	Ki	=	88.00	7.06	-15	7	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	334.1	3	4	9	-1.30	Nc1ncnc2c1ncn2[C@@H]1O[C@H](C(=O)NC2CCC2)[C@@H](O)[C@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL2070508	76963	None	2	Rat	Binding	Ki	=	49.00	7.31	-1	7	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	348.2	3	4	9	-0.91	Nc1ncnc2c1ncn2[C@@H]1O[C@H](C(=O)NC2CCCC2)[C@@H](O)[C@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL2092773	77839	None	0	Rat	Binding	Ki	=	55.60	7.25	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	376.2	3	4	9	-0.28	C[C@H]1CC[C@@H](NC(=O)[C@H]2O[C@@H](n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)CC1	https://dx.doi.org/10.1021/jm000150k
CHEMBL2092859	77849	None	0	Rat	Binding	Ki	=	12.90	7.89	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	376.2	3	4	9	-0.28	C[C@H]1CC[C@H](NC(=O)[C@H]2O[C@@H](n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)CC1	https://dx.doi.org/10.1021/jm000150k
CHEMBL2113434	79263	None	1	Rat	Binding	Ki	=	58.00	7.24	1	5	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	310.1	3	4	10	-2.29	CONC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL2113436	79265	None	0	Rat	Binding	Ki	=	6850.00	5.16	-5	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	336.2	2	4	9	-1.06	CC(C)(C)NC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL2113489	79318	None	0	Rat	Binding	Ki	=	18.00	7.75	141	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	362.2	3	4	9	-0.52	Nc1ncnc2c1ncn2[C@@H]1O[C@H](C(=O)NC2CCCCC2)[C@@H](O)[C@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL2113492	79321	None	0	Rat	Binding	Ki	=	12.00	7.92	50	4	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	350.2	6	4	9	-0.67	CCCCCNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL261482	96386	None	27	Rat	Binding	Ki	=	96.00	7.02	-50	10	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	320.1	3	4	9	-1.69	Nc1ncnc2c1ncn2[C@@H]1O[C@H](C(=O)NC2CC2)[C@@H](O)[C@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL519809	191890	None	12	Rat	Binding	Ki	=	51.00	7.29	-4	8	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	294.1	2	4	9	-2.23	CNC(=O)[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL605866	204079	None	0	Rat	Binding	Ki	=	64.00	7.19	1	3	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	280.1	2	4	9	-2.49	NC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL607717	204394	None	0	Rat	Binding	Ki	=	42.00	7.38	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	370.1	4	4	9	-0.66	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NCc2ccccc2)[C@@H](O)[C@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL607719	204395	None	0	Rat	Binding	Ki	=	19.00	7.72	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	364.2	7	4	9	-0.28	CCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL608000	204431	None	0	Rat	Binding	Ki	=	1040.00	5.98	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	414.2	3	4	9	0.11	Nc1ncnc2c1ncn2C1O[C@H](C(=O)NC23CC4CC(CC(C4)C2)C3)[C@@H](O)[C@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL608003	204432	None	0	Rat	Binding	Ki	=	140.00	6.85	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	430.2	6	4	11	-0.64	COc1ccc(CNC(=O)[C@H]2OC(n3cnc4c(N)ncnc43)[C@H](O)[C@@H]2O)cc1OC	https://dx.doi.org/10.1021/jm000150k
CHEMBL608293	204471	None	0	Rat	Binding	Ki	=	20.00	7.70	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	352.1	5	4	10	-1.27	CC(C)CONC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k
CHEMBL608296	204472	None	0	Rat	Binding	Ki	=	21.00	7.68	-	1	Binding activity of P3 purinoceptor-like protein (P3LP) using radioligand 40 nM [3H]NECA from rat brain membranes	ChEMBL	392.2	9	4	9	0.50	CCCCCCCCNC(=O)[C@H]1OC(n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O	https://dx.doi.org/10.1021/jm000150k

Showing 1 to 20 of 41 entries

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

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Ligand source activities (1 row/activity)