Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
| 131648253 | 3039 | None | 0 | Mouse | Functional | pEC50 | = | 10.7 | 10.7 | - | 1 | High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83 |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
| 155817507 | 3039 | None | 0 | Mouse | Functional | pEC50 | = | 10.7 | 10.7 | - | 1 | High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83 |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
| 9139 | 3039 | None | 0 | Mouse | Functional | pEC50 | = | 10.7 | 10.7 | - | 1 | High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83 |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
| 131648253 | 3039 | None | 0 | Mouse | Functional | pEC50 | = | 7.0 | 7.0 | - | 1 | Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83 |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
| 155817507 | 3039 | None | 0 | Mouse | Functional | pEC50 | = | 7.0 | 7.0 | - | 1 | Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83 |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
| 9139 | 3039 | None | 0 | Mouse | Functional | pEC50 | = | 7.0 | 7.0 | - | 1 | Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83 |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
| 32051 | 4151 | None | 0 | Mouse | Functional | pEC50 | = | 5 | 5.0 | - | 1 | UnclassifiedUnclassified |
Guide to Pharmacology | 64 | 0 | 0 | 0 | -0.0 | [Zn+2] | 23335960 | ||
| 566 | 4151 | None | 0 | Mouse | Functional | pEC50 | = | 5 | 5.0 | - | 1 | UnclassifiedUnclassified |
Guide to Pharmacology | 64 | 0 | 0 | 0 | -0.0 | [Zn+2] | 23335960 | ||
Showing 1 to 8 of 8 entries
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
| 9140 | 3040 | None | 0 | Mouse | Binding | pKd | = | 8.1 | 8.1 | - | 1 | N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations. |
Guide to Pharmacology | None | None | None | None | 27117253 | ||||
Showing 1 to 1 of 1 entries