Ligand source activities (1 row/activity)
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 2365 | 7390 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 239 | 7390 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 4755801 | 7390 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| CHEMBL297569 | 7390 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| DB03107 | 7390 | 0 | None | -3 | 3 | Mouse | 4.4 | pEC50 | = | 4.4 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 2365 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 2365 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| 239 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 239 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| 4755801 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 4755801 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| CHEMBL297569 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| CHEMBL297569 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| DB03107 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| DB03107 | 7390 | 0 | None | -1 | 3 | Human | 4.8 | pEC50 | = | 4.8 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 23396314 | ||
| 2365 | 7390 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 239 | 7390 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| 4755801 | 7390 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| CHEMBL297569 | 7390 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| DB03107 | 7390 | 0 | None | 1 | 3 | Rat | 4.9 | pEC50 | = | 4.9 | Functional | Guide to Pharmacology | 89 | 2 | 2 | 2 | -0.6 | NCCC(=O)O | 15037633 | ||
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |