Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
| 10321 | 1705 | None | 0 | Human | Functional | pEC50 | = | 6.4 | 6.4 | - | 1 | In a TCF/LEF reporter assay with WRE-GFP constructs.In a TCF/LEF reporter assay with WRE-GFP constructs. |
Guide to Pharmacology | 322 | 3 | 4 | 3 | 3.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O | 29293331 | ||
| 137553171 | 1705 | None | 0 | Human | Functional | pEC50 | = | 6.4 | 6.4 | - | 1 | In a TCF/LEF reporter assay with WRE-GFP constructs.In a TCF/LEF reporter assay with WRE-GFP constructs. |
Guide to Pharmacology | 322 | 3 | 4 | 3 | 3.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O | 29293331 | ||
| 10321 | 1705 | None | 0 | Human | Functional | pIC50 | = | 6.7 | 6.7 | - | 1 | In TCF/LEF reporter assays with WRE-GFP constructsIn TCF/LEF reporter assays with WRE-GFP constructs |
Guide to Pharmacology | 322 | 3 | 4 | 3 | 3.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O | 25751279 | ||
| 137553171 | 1705 | None | 0 | Human | Functional | pIC50 | = | 6.7 | 6.7 | - | 1 | In TCF/LEF reporter assays with WRE-GFP constructsIn TCF/LEF reporter assays with WRE-GFP constructs |
Guide to Pharmacology | 322 | 3 | 4 | 3 | 3.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O | 25751279 | ||
| 10322 | 1704 | None | 0 | Human | Functional | pIC50 | = | 6.2 | 6.2 | - | 1 | In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs. |
Guide to Pharmacology | 360 | 3 | 3 | 3 | 5.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 | 25751279 | ||
| 10322 | 1704 | None | 0 | Human | Functional | pIC50 | = | 6.2 | 6.2 | - | 1 | In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs. |
Guide to Pharmacology | 360 | 3 | 3 | 3 | 5.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 | 29293331 | ||
| 90478321 | 1704 | None | 0 | Human | Functional | pIC50 | = | 6.2 | 6.2 | - | 1 | In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs. |
Guide to Pharmacology | 360 | 3 | 3 | 3 | 5.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 | 25751279 | ||
| 90478321 | 1704 | None | 0 | Human | Functional | pIC50 | = | 6.2 | 6.2 | - | 1 | In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs. |
Guide to Pharmacology | 360 | 3 | 3 | 3 | 5.9 | O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 | 29293331 | ||
Showing 1 to 8 of 8 entries
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
| 2947 | 2865 | None | 0 | Mouse | Binding | pKd | None | 8.4 | 8.4 | - | 1 | UnclassifiedUnclassified |
Guide to Pharmacology | None | None | None | None | 15035989 | ||||
Showing 1 to 1 of 1 entries