Ligand source activities (1 row/activity)



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Ligands Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb ID #Vendors Reference
ligand		 Fold selectivity
(Potency)		 # tested GPCRs
(Potency)		 Species p-value
(-log)		 Type Activity
Relation		 Activity
Value		 Assay Type Assay Description Source Mol
weight		 Rot
Bonds		 H don H acc LogP Smiles DOI
10321 8486 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
In a TCF/LEF reporter assay with WRE-GFP constructs.In a TCF/LEF reporter assay with WRE-GFP constructs.
Guide to Pharmacology 322 3 4 3 3.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O 29293331
137553171 8486 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
In a TCF/LEF reporter assay with WRE-GFP constructs.In a TCF/LEF reporter assay with WRE-GFP constructs.
Guide to Pharmacology 322 3 4 3 3.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O 29293331
10321 8486 0 None - 1 Human 6.7 pIC50 = 6.7 Functional
In TCF/LEF reporter assays with WRE-GFP constructsIn TCF/LEF reporter assays with WRE-GFP constructs
Guide to Pharmacology 322 3 4 3 3.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O 25751279
137553171 8486 0 None - 1 Human 6.7 pIC50 = 6.7 Functional
In TCF/LEF reporter assays with WRE-GFP constructsIn TCF/LEF reporter assays with WRE-GFP constructs
Guide to Pharmacology 322 3 4 3 3.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)C(=O)O 25751279
10322 8485 0 None - 1 Human 6.2 pIC50 = 6.2 Functional
In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.
Guide to Pharmacology 360 3 3 3 5.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 25751279
10322 8485 0 None - 1 Human 6.2 pIC50 = 6.2 Functional
In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.
Guide to Pharmacology 360 3 3 3 5.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 29293331
90478321 8485 0 None - 1 Human 6.2 pIC50 = 6.2 Functional
In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.
Guide to Pharmacology 360 3 3 3 5.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 25751279
90478321 8485 0 None - 1 Human 6.2 pIC50 = 6.2 Functional
In TCF/LEF reporter assays with WRE-GFP constructs.In TCF/LEF reporter assays with WRE-GFP constructs.
Guide to Pharmacology 360 3 3 3 5.9 O=C(Nc1ccc2c(c1)cccc2)Nc1cc(O)cc(c1)c1cccs1 29293331


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Ligands Receptor Assay information Chemical information
Sel. page Common
name		 GPCRdb ID #Vendors Reference
ligand		 Fold selectivity
(Affinity)		 # tested GPCRs
(Affinity)		 Species p-value
(-log)		 Type Activity
Relation		 Activity
Value		 Assay Type Assay Description Source Mol
weight		 Rot
Bonds		 H don H acc LogP Smiles DOI
2947 9640 0 None - 1 Mouse 8.4 pKd None 8.4 Binding
UnclassifiedUnclassified
Guide to Pharmacology None None None None 15035989