GPCRdb

Ligand source activities (1 row/activity)

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	165271	105532	33	None	-	1	Human	10.5	pEC50	=	10.5	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	141	3	3	3	-0.7	N[C@H](CO)Cc1c[nH]cn1	nan
	CHEMBL278081	105532	33	None	-	1	Human	10.5	pEC50	=	10.5	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	141	3	3	3	-0.7	N[C@H](CO)Cc1c[nH]cn1	nan
	CHEMBL4517318	220750	68	None	-	1	Human	9.8	pEC50	=	9.8	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43CO)[C@@H]1CCC2=O	nan
	70914	23248	99	None	-	1	Human	9.6	pEC50	=	9.6	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	189	5	3	3	-0.6	CC(=O)N[C@@H](CCC(=O)O)C(=O)O	nan
	CHEMBL1234751	23248	99	None	-	1	Human	9.6	pEC50	=	9.6	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	189	5	3	3	-0.6	CC(=O)N[C@@H](CCC(=O)O)C(=O)O	nan
	440832	20878	8	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	271	1	4	4	3.2	Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1	nan
	CHEMBL1197905	20878	8	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	271	1	4	4	3.2	Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1	nan
	CHEMBL591036	20878	8	None	-	1	Human	9.4	pEC50	=	9.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	271	1	4	4	3.2	Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1	nan
	10204	78242	27	None	-	1	Human	9.2	pEC50	=	9.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	288	0	1	2	3.9	C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]1CC[C@H]2O	nan
	CHEMBL196228	78242	27	None	-	1	Human	9.2	pEC50	=	9.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	288	0	1	2	3.9	C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]1CC[C@H]2O	nan
	222865	23169	31	None	-	1	Human	9.1	pEC50	=	9.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	288	0	0	2	4.2	C[C@]12CCC(=O)C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12	nan
	CHEMBL1230438	23169	31	None	-	1	Human	9.1	pEC50	=	9.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	288	0	0	2	4.2	C[C@]12CCC(=O)C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12	nan
	3812	7504	42	None	-2	3	Human	8.9	pEC50	=	8.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		None	nan
	439201	7504	42	None	-2	3	Human	8.9	pEC50	=	8.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		None	nan
	649	7504	42	None	-2	3	Human	8.9	pEC50	=	8.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		None	nan
	CHEMBL406291	7504	42	None	-2	3	Human	8.9	pEC50	=	8.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		None	nan
	DB12126	7504	42	None	-2	3	Human	8.9	pEC50	=	8.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		None	nan
	12025	105370	89	None	-	1	Human	8.7	pEC50	=	8.7	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	85	0	1	1	-0.1	O=C1CCCN1	nan
	CHEMBL276849	105370	89	None	-	1	Human	8.7	pEC50	=	8.7	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	85	0	1	1	-0.1	O=C1CCCN1	nan
	CHEMBL4556656	220785	44	None	-	1	Human	8.7	pEC50	=	8.7	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		O=C(O)[C@@H](O)CO	nan
	CHEMBL4590792	220798	38	None	-	1	Human	6.0	pEC50	=	6	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		O=C[C@H](O[C@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@@H](O)[C@H](O)[C@H](O)CO	nan
	11163	107478	113	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	132	3	3	3	-1.9	NCC(=O)NCC(=O)O	nan
	1548897	107478	113	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	132	3	3	3	-1.9	NCC(=O)NCC(=O)O	nan
	CHEMBL292467	107478	113	None	-	1	Human	5.0	pEC50	=	5.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	132	3	3	3	-1.9	NCC(=O)NCC(=O)O	nan
	171161	74063	49	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	264	7	2	4	1.0	COc1ccc(NC=O)c(C(=O)CCNC(C)=O)c1	nan
	CHEMBL1882218	74063	49	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	264	7	2	4	1.0	COc1ccc(NC=O)c(C(=O)CCNC(C)=O)c1	nan
	5460362	108475	66	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	160	3	3	3	-1.1	C[C@@H](N)C(=O)N[C@H](C)C(=O)O	nan
	6992112	108475	66	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	160	3	3	3	-1.1	C[C@@H](N)C(=O)N[C@H](C)C(=O)O	nan
	CHEMBL299420	108475	66	None	-	1	Human	4.9	pEC50	=	4.9	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	160	3	3	3	-1.1	C[C@@H](N)C(=O)N[C@H](C)C(=O)O	nan
	1176	214988	97	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	60	0	2	1	-1.0	NC(N)=O	nan
	CHEMBL985	214988	97	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	60	0	2	1	-1.0	NC(N)=O	nan
	CHEMBL4574750	220795	18	None	-	1	Human	7.6	pEC50	=	7.6	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		Nc1ncnc2c1ncn2C1OC(CO)C2OP(=O)(O)OC21	nan
	964	23163	42	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	104	2	2	3	-1.4	O=C(O)C(=O)CO	nan
	CHEMBL1230192	23163	42	None	-	1	Human	6.4	pEC50	=	6.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	104	2	2	3	-1.4	O=C(O)C(=O)CO	nan
	3636	7149	125	None	22908	2	Human	8.3	pEC50	=	8.3	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	nan
	51	7149	125	None	22908	2	Human	8.3	pEC50	=	8.3	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	nan
	CHEMBL1686	7149	125	None	22908	2	Human	8.3	pEC50	=	8.3	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	nan
	DB08845	7149	125	None	22908	2	Human	8.3	pEC50	=	8.3	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	146	4	2	3	-0.5	OC(=O)CCC(=O)C(=O)O	nan
	5756	76402	77	None	-	1	Human	4.3	pEC50	=	4.3	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	288	0	3	3	2.6	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O	nan
	CHEMBL193482	76402	77	None	-	1	Human	4.3	pEC50	=	4.3	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	288	0	3	3	2.6	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O	nan
	124072	114312	88	None	-	1	Human	6.2	pEC50	=	6.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	372	10	2	6	3.2	COc1cc(CCC(=O)CC(=O)CCc2ccc(O)c(OC)c2)ccc1O	nan
	CHEMBL318743	114312	88	None	-	1	Human	6.2	pEC50	=	6.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	372	10	2	6	3.2	COc1cc(CCC(=O)CC(=O)CCc2ccc(O)c(OC)c2)ccc1O	nan
	1319	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	4084	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	4635	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	5257127	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	727	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	750	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	CHEMBL773	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	DB00145	8607	130	None	12302	2	Human	7.2	pEC50	=	7.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	75	1	2	2	-1.0	NCC(=O)O	nan
	CHEMBL4566376	220792	0	None	-	1	Human	8.2	pEC50	=	8.2	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL		None	None	None		None	nan
	1055	9768	105	None	2884	2	Human	8.0	pEC50	=	8.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	256	14	1	1	5.6	CCCCCCCCCCCCCCCC(=O)O	nan
	135369651	9768	105	None	2884	2	Human	8.0	pEC50	=	8.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	256	14	1	1	5.6	CCCCCCCCCCCCCCCC(=O)O	nan
	985	9768	105	None	2884	2	Human	8.0	pEC50	=	8.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	256	14	1	1	5.6	CCCCCCCCCCCCCCCC(=O)O	nan
	CHEMBL82293	9768	105	None	2884	2	Human	8.0	pEC50	=	8.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	256	14	1	1	5.6	CCCCCCCCCCCCCCCC(=O)O	nan
	DB03796	9768	105	None	2884	2	Human	8.0	pEC50	=	8.0	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	256	14	1	1	5.6	CCCCCCCCCCCCCCCC(=O)O	nan
	5282379	201763	69	None	25	4	Human	6.8	pIC50	=	6.8	Functional	Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	300	5	1	1	5.6	CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1	nan
	CHEMBL547	201763	69	None	25	4	Human	6.8	pIC50	=	6.8	Functional	Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	ChEMBL	300	5	1	1	5.6	CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1	nan
	5756	76402	77	None	-	1	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	288	0	3	3	2.6	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O	None
	CHEMBL193482	76402	77	None	-	1	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	288	0	3	3	2.6	C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O	None
	10577	224487	0	None	-	1	Human	8.4	pEC50	=	8.4	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	488	8	3	7	3.4	C[C@]12CC[C@H]3[C@@H](CCC4=CC(O)=CC=C34)[C@@H]1C[C@@H](OC(=O)CCC(O)=O)[C@@H]2OC(=O)CCC(O)=O	None
	1319	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	4084	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	4635	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	5257127	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	727	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	750	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	CHEMBL773	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	DB00145	8607	130	None	12302	2	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	75	1	2	2	-1.0	NCC(=O)O	None
	1176	214988	97	None	-	1	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	60	0	2	1	-1.0	NC(N)=O	None
	CHEMBL985	214988	97	None	-	1	Human	8.1	pEC50	=	8.1	Functional	Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	60	0	2	1	-1.0	NC(N)=O	None
	5282379	201763	69	None	25	4	Human	8.2	pIC50	=	8.2	Functional	Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	300	5	1	1	5.6	CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1	None
	CHEMBL547	201763	69	None	25	4	Human	8.2	pIC50	=	8.2	Functional	Antagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAntagonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay	Drug Central	300	5	1	1	5.6	CC1=C(/C=C/C(C)=C/C=C/C(C)=C\C(=O)O)C(C)(C)CCC1	None

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

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Ligand source activities (1 row/activity)