Ligand source activities (1 row/activity)
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
| |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
| 165271 | 98810 | None | 22 | Human | Functional | pEC50 | = | 10.5 | 10.5 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 141 | 3 | 3 | 3 | -0.7 | N[C@H](CO)Cc1c[nH]cn1 | nan | ||
| CHEMBL278081 | 98810 | None | 22 | Human | Functional | pEC50 | = | 10.5 | 10.5 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 141 | 3 | 3 | 3 | -0.7 | N[C@H](CO)Cc1c[nH]cn1 | nan | ||
| CHEMBL4517318 | 216434 | None | 43 | Human | Functional | pEC50 | = | 9.8 | 9.8 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43CO)[C@@H]1CCC2=O | nan | ||||
| 70914 | 16483 | None | 57 | Human | Functional | pEC50 | = | 9.6 | 9.6 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 189 | 5 | 3 | 3 | -0.6 | CC(=O)N[C@@H](CCC(=O)O)C(=O)O | nan | ||
| CHEMBL1234751 | 16483 | None | 57 | Human | Functional | pEC50 | = | 9.6 | 9.6 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 189 | 5 | 3 | 3 | -0.6 | CC(=O)N[C@@H](CCC(=O)O)C(=O)O | nan | ||
| 440832 | 14111 | None | 3 | Human | Functional | pEC50 | = | 9.4 | 9.4 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 271 | 1 | 4 | 4 | 3.2 | Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1 | nan | ||
| CHEMBL1197905 | 14111 | None | 3 | Human | Functional | pEC50 | = | 9.4 | 9.4 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 271 | 1 | 4 | 4 | 3.2 | Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1 | nan | ||
| CHEMBL591036 | 14111 | None | 3 | Human | Functional | pEC50 | = | 9.4 | 9.4 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 271 | 1 | 4 | 4 | 3.2 | Oc1ccc(-c2[o+]c3cc(O)cc(O)c3cc2O)cc1 | nan | ||
| 10204 | 71491 | None | 14 | Human | Functional | pEC50 | = | 9.2 | 9.2 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 288 | 0 | 1 | 2 | 3.9 | C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]1CC[C@H]2O | nan | ||
| CHEMBL196228 | 71491 | None | 14 | Human | Functional | pEC50 | = | 9.2 | 9.2 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 288 | 0 | 1 | 2 | 3.9 | C[C@]12CC[C@H]3[C@@H](CCC4=CC(=O)CC[C@@]43C)[C@@H]1CC[C@H]2O | nan | ||
| 222865 | 16404 | None | 16 | Human | Functional | pEC50 | = | 9.1 | 9.1 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 288 | 0 | 0 | 2 | 4.2 | C[C@]12CCC(=O)C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12 | nan | ||
| CHEMBL1230438 | 16404 | None | 16 | Human | Functional | pEC50 | = | 9.1 | 9.1 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 288 | 0 | 0 | 2 | 4.2 | C[C@]12CCC(=O)C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)C(=O)CC[C@@H]12 | nan | ||
| 3812 | 717 | None | 37 | Human | Functional | pEC50 | = | 8.9 | 8.9 | -2 | 3 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | None | nan | ||||
| 439201 | 717 | None | 37 | Human | Functional | pEC50 | = | 8.9 | 8.9 | -2 | 3 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | None | nan | ||||
| 649 | 717 | None | 37 | Human | Functional | pEC50 | = | 8.9 | 8.9 | -2 | 3 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | None | nan | ||||
| CHEMBL406291 | 717 | None | 37 | Human | Functional | pEC50 | = | 8.9 | 8.9 | -2 | 3 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | None | nan | ||||
| DB12126 | 717 | None | 37 | Human | Functional | pEC50 | = | 8.9 | 8.9 | -2 | 3 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | None | nan | ||||
| 12025 | 98647 | None | 55 | Human | Functional | pEC50 | = | 8.7 | 8.7 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 85 | 0 | 1 | 1 | -0.1 | O=C1CCCN1 | nan | ||
| CHEMBL276849 | 98647 | None | 55 | Human | Functional | pEC50 | = | 8.7 | 8.7 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 85 | 0 | 1 | 1 | -0.1 | O=C1CCCN1 | nan | ||
| CHEMBL4556656 | 216477 | None | 35 | Human | Functional | pEC50 | = | 8.7 | 8.7 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | O=C(O)[C@@H](O)CO | nan | ||||
| CHEMBL4590792 | 216499 | None | 34 | Human | Functional | pEC50 | = | 6 | 6.0 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | O=C[C@H](O[C@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)[C@@H](O)[C@H](O)[C@H](O)CO | nan | ||||
| 11163 | 100756 | None | 67 | Human | Functional | pEC50 | = | 5.0 | 5.0 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 132 | 3 | 3 | 3 | -1.9 | NCC(=O)NCC(=O)O | nan | ||
| 1548897 | 100756 | None | 67 | Human | Functional | pEC50 | = | 5.0 | 5.0 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 132 | 3 | 3 | 3 | -1.9 | NCC(=O)NCC(=O)O | nan | ||
| CHEMBL292467 | 100756 | None | 67 | Human | Functional | pEC50 | = | 5.0 | 5.0 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 132 | 3 | 3 | 3 | -1.9 | NCC(=O)NCC(=O)O | nan | ||
| 171161 | 67310 | None | 39 | Human | Functional | pEC50 | = | 4.9 | 4.9 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 264 | 7 | 2 | 4 | 1.0 | COc1ccc(NC=O)c(C(=O)CCNC(C)=O)c1 | nan | ||
| CHEMBL1882218 | 67310 | None | 39 | Human | Functional | pEC50 | = | 4.9 | 4.9 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 264 | 7 | 2 | 4 | 1.0 | COc1ccc(NC=O)c(C(=O)CCNC(C)=O)c1 | nan | ||
| 5460362 | 101753 | None | 42 | Human | Functional | pEC50 | = | 4.9 | 4.9 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 160 | 3 | 3 | 3 | -1.1 | C[C@@H](N)C(=O)N[C@H](C)C(=O)O | nan | ||
| 6992112 | 101753 | None | 42 | Human | Functional | pEC50 | = | 4.9 | 4.9 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 160 | 3 | 3 | 3 | -1.1 | C[C@@H](N)C(=O)N[C@H](C)C(=O)O | nan | ||
| CHEMBL299420 | 101753 | None | 42 | Human | Functional | pEC50 | = | 4.9 | 4.9 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 160 | 3 | 3 | 3 | -1.1 | C[C@@H](N)C(=O)N[C@H](C)C(=O)O | nan | ||
| 1176 | 210668 | None | 62 | Human | Functional | pEC50 | = | 7.6 | 7.6 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 60 | 0 | 2 | 1 | -1.0 | NC(N)=O | nan | ||
| CHEMBL985 | 210668 | None | 62 | Human | Functional | pEC50 | = | 7.6 | 7.6 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 60 | 0 | 2 | 1 | -1.0 | NC(N)=O | nan | ||
| CHEMBL4574750 | 216490 | None | 13 | Human | Functional | pEC50 | = | 7.6 | 7.6 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | None | None | None | Nc1ncnc2c1ncn2C1OC(CO)C2OP(=O)(O)OC21 | nan | ||||
| 964 | 16398 | None | 30 | Human | Functional | pEC50 | = | 6.4 | 6.4 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 104 | 2 | 2 | 3 | -1.4 | O=C(O)C(=O)CO | nan | ||
| CHEMBL1230192 | 16398 | None | 30 | Human | Functional | pEC50 | = | 6.4 | 6.4 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 104 | 2 | 2 | 3 | -1.4 | O=C(O)C(=O)CO | nan | ||
| 3636 | 361 | None | 69 | Human | Functional | pEC50 | = | 8.3 | 8.3 | 22908 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 146 | 4 | 2 | 3 | -0.5 | OC(=O)CCC(=O)C(=O)O | nan | ||
| 51 | 361 | None | 69 | Human | Functional | pEC50 | = | 8.3 | 8.3 | 22908 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 146 | 4 | 2 | 3 | -0.5 | OC(=O)CCC(=O)C(=O)O | nan | ||
| CHEMBL1686 | 361 | None | 69 | Human | Functional | pEC50 | = | 8.3 | 8.3 | 22908 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 146 | 4 | 2 | 3 | -0.5 | OC(=O)CCC(=O)C(=O)O | nan | ||
| DB08845 | 361 | None | 69 | Human | Functional | pEC50 | = | 8.3 | 8.3 | 22908 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 146 | 4 | 2 | 3 | -0.5 | OC(=O)CCC(=O)C(=O)O | nan | ||
| 5756 | 69649 | None | 49 | Human | Functional | pEC50 | = | 4.3 | 4.3 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 288 | 0 | 3 | 3 | 2.6 | C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O | nan | ||
| CHEMBL193482 | 69649 | None | 49 | Human | Functional | pEC50 | = | 4.3 | 4.3 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 288 | 0 | 3 | 3 | 2.6 | C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1C[C@@H](O)[C@@H]2O | nan | ||
| 124072 | 107591 | None | 60 | Human | Functional | pEC50 | = | 6.2 | 6.2 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 372 | 10 | 2 | 6 | 3.2 | COc1cc(CCC(=O)CC(=O)CCc2ccc(O)c(OC)c2)ccc1O | nan | ||
| CHEMBL318743 | 107591 | None | 60 | Human | Functional | pEC50 | = | 6.2 | 6.2 | - | 1 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 372 | 10 | 2 | 6 | 3.2 | COc1cc(CCC(=O)CC(=O)CCc2ccc(O)c(OC)c2)ccc1O | nan | ||
| 1319 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| 4084 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| 4635 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| 5257127 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| 727 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| 750 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| CHEMBL773 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
| DB00145 | 1826 | None | 72 | Human | Functional | pEC50 | = | 7.2 | 7.2 | 12302 | 2 | Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assayAgonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay |
ChEMBL | 75 | 1 | 2 | 2 | -1.0 | NCC(=O)O | nan | ||
Showing 1 to 50 of 73 entries
| Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
Ligands (move mouse cursor over ligand name to see structure)
| Receptor
| Activity
| Chemical information
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|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name
| GPCRdb ID
| Reference ligand
| Vendors | Species
| Assay Type
| Activity Type
| Activity Relation
| Activity Value | p-value (-log) | Fold selectivity | Tested GPCRs | Assay Description
| Source
| Mol weight | Rot Bonds | H don | H acc | LogP | Smiles
| DOI
| |
| No data available in table | ||||||||||||||||||||||
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