GPCRdb

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Ligand source activities (1 row/activity)

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	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

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	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

	Ligands				Receptor	Activity									Chemical information
	Common name	GPCRdb ID	Reference ligand	Vendors	Species	Assay Type	Activity Type	Activity Relation	Activity Value	p-value (-log)	Fold selectivity	Tested GPCRs	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI

	abscisic acid	227	None	44	Human	Functional	pIC50	=	-	4.46	-1096	5	Unclassified	Guide to Pharmacology	264.1	3	2	3	2.25	CC1=CC(=O)CC(C)(C)C1(O)/C=C/C(C)=C\C(=O)O	https://pubmed.ncbi.nlm.nih.gov/25844797
	azithromycin	561	None	43	Human	Functional	pEC50	=	-	4.13	-562	3	Unclassified	Guide to Pharmacology	748.5	7	5	14	1.90	CC[C@H]1OC(=O)[C@H](C)[C@@H](O[C@H]2C[C@@](C)(OC)[C@@H](O)[C@H](C)O2)[C@H](C)[C@@H](O[C@@H]2O[C@H](C)C[C@H](N(C)C)[C@H]2O)[C@](C)(O)C[C@@H](C)CN(C)[C@H](C)[C@@H](O)[C@]1(C)O	https://pubmed.ncbi.nlm.nih.gov/30011231
	colchicine	964	None	47	Human	Functional	pEC50	=	-	2.99	-1148	6	Unclassified	Guide to Pharmacology	399.2	5	1	6	2.87	COc1cc2c(c(OC)c1OC)-c1ccc(OC)c(=O)cc1[C@@H](NC(C)=O)CC2	https://pubmed.ncbi.nlm.nih.gov/20022913
	isoprenaline	2091	None	34	Human	Functional	pEC50	=	8.31	8.08	-63	49	Agonist activity at human TAS2R4 expressed in HEK293T cells co-expressing Galpha15 assessed as increase in intracellular calcium level by Calcium-3 dye based fluorescence assay	Drug Central	211.1	4	4	4	1.13	CC(C)NCC(O)c1ccc(O)c(O)c1	-
	isoprenaline	2091	None	34	Human	Functional	EC50	=	4.90	8.31	-63	49	Agonist activity at human TAS2R4 expressed in HEK293T cells co-expressing Galpha15 assessed as increase in intracellular calcium level by Calcium-3 dye based fluorescence assay	ChEMBL	211.1	4	4	4	1.13	CC(C)NCC(O)c1ccc(O)c(O)c1	-
	L-Trp-Trp-Trp	2372	None	0	Human	Functional	pEC50	=	-	4.52	-	5	Unclassified	Guide to Pharmacology	-	-	-	-	-	-	https://pubmed.ncbi.nlm.nih.gov/23214402
	stevioside	3692	None	0	Human	Functional	pEC50	=	-	3.47	-	1	Unclassified	Guide to Pharmacology	804.4	9	11	18	-2.94	C=C1C[C@@]23CC[C@H]4[C@@](C)(CCC[C@@]4(C)C(=O)O[C@@H]4O[C@H](CO)[C@@H](O)[C@H](O)[C@H]4O)[C@@H]2CC[C@]1(O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O)C3	https://pubmed.ncbi.nlm.nih.gov/22616809

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