Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
aa2br_rat 326 C-term S => A N/A N/A Matharu AL et al (2001)
aa2br_rat 329 C-term S => G N/A N/A Matharu AL et al (2001)
aa2br_rat 329 C-term S => A 2.273↓ EC50 (Functional - cAMP accumulation) NECA Matharu AL et al (2001) Jespers W et al (2018)
aa2br_rat 329 C-term S => G 1.467↑ EC50 (Functional - cAMP accumulation) NECA Matharu AL et al (2001) Jespers W et al (2018)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 S A L Q ICL1ECL1 F C T ECL1ICL2 P L R Y K G L V ICL2ECL2 W N S K D R A T S N C T E P G D G I T N K S C C P V K C L F E N V V ECL2ICL3 L M E ICL3ECL3 P A L A K D K ECL3N-term M Q L N-termC-term G G S G Q A G G Q S T F S L S L C-term E T Q D A L Y V A L E L V I A A L A V A G N V L V C A A V G A S T P T N Y F L V S L A T A D V A V G L F A I P F A I T I S L G D F H S C L F L A C F V L V L T Q S S I F S L L A V A V D R Y L A I R V T G T R A R G I I A V L W V L A F G I G L T P F L G P M S Y M V Y F N F F G C V L P P L L I M M V I Y I K I F M V A C K Q L Q H M E H S R T T L Q R E I H A A K S L A M I V G I F A L C W L P V H A I N C I T L F H P K W V M N V A I L L S H A N S V V N P I V Y A Y R N R D F H R Y V L T K F R Y S I I S R C Q T D
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
V N G A V A L A A I V L E L A V Y L A D 1 V S L A T A D V A V G F L A I P F A I T I 2 A L L S F I S S Q T L V L V F C A L F L 3 A R G I I A V L W V L A F G I G L T P F 4 Y I V M M I L L P P L V C G F F N F Y V M Y 5 A M I V G I F A L C W L P V H A I N C I 6 I P N V V S N A H S L L I A V N M V W 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
A2B receptor