Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
adrb2_human 12.50x50 64 ICL1 L => G N/A N/A O'Dowd BF et al (1988)
adrb2_human 2.48x48 77 TM2 C => S N/A N/A Fraser CM et al (1989)
adrb2_human 2.50x50 79 TM2 D => N N/A N/A Chung FZ et al (1988)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Fraser CM et al (1988)
adrb2_human 34.50x50 138 ICL2 P => S N/A N/A O'Dowd BF et al (1988)
adrb2_human 4.56x56 164 TM4 T => I N/A N/A Green SA et al (1993)
adrb2_human 6.30x30 268 TM6 E => G N/A N/A O'Dowd BF et al (1988)
adrb2_human 6.47x47 285 TM6 C => S N/A N/A Fraser CM et al (1989)
adrb2_human 7.39x38 312 TM7 N => F N/A N/A Suryanarayana S et al (1993)
adrb2_human 7.39x38 312 TM7 N => A N/A N/A Suryanarayana S et al (1993)
adrb2_human 7.39x38 312 TM7 N => T N/A N/A Suryanarayana S et al (1993)
adrb2_human 7.39x38 312 TM7 N => Q N/A N/A Suryanarayana S et al (1993)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Barak LS et al (1994)
adrb2_human 7.54x54 327 TM7 C => S N/A N/A Fraser CM et al (1989)
adrb2_human 7.54x54 327 TM7 C => R N/A N/A O'Dowd BF et al (1988)
adrb2_human 8.59x59 341 H8 C => G N/A N/A O'Dowd BF et al (1988)
adrb2_human 8.59x59 341 H8 C => G N/A N/A O'Dowd BF et al (1989)
adrb2_human 350 C-term Y => A N/A N/A Valiquette M et al (1993)
adrb2_human 354 C-term Y => A N/A N/A Valiquette M et al (1993)
adrb2_human 184 ECL2 C => V N/A N/A Liggett SB et al (1989)
adrb2_human 8.59x59 341 H8 C => G N/A N/A Moffett S et al (1993)
adrb2_human 2.48x48 77 TM2 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 3.25x25 106 TM3 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 3.35x35 116 TM3 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 3.44x44 125 TM3 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 184 ECL2 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 190 ECL2 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 45.50x50 191 ECL2 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 6.47x47 285 TM6 C => V N/A N/A Dohlman HG et al (1990)
adrb2_human 8.59x59 341 H8 C => G N/A N/A Campbell PT et al (1991)
adrb2_human 7.49x49 322 TM7 N => A N/A N/A Barak LS et al (1995)
adrb2_human 7.49x49 322 TM7 N => D N/A N/A Barak LS et al (1995)
adrb2_human 7.50x50 323 TM7 P => A N/A N/A Barak LS et al (1995)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Barak LS et al (1995)
adrb2_human 7.53x53 326 TM7 Y => F N/A N/A Barak LS et al (1995)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Menard L et al (1996)
adrb2_human 7.37x36 310 TM7 L => F N/A N/A Mizobe T et al (1996)
adrb2_human 7.38x37 311 TM7 L => F N/A N/A Mizobe T et al (1996)
adrb2_human 7.39x38 312 TM7 N => F N/A N/A Mizobe T et al (1996)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Ferguson SS et al (1995)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Ferguson SS et al (1996)
adrb2_human 7.39x38 312 TM7 N => F N/A N/A Suryanarayana S et al (1991)
adrb2_human 34.53x53 141 ICL2 Y => F N/A N/A Valiquette M et al (1995)
adrb2_human 350 C-term Y => A N/A N/A Valiquette M et al (1995)
adrb2_human 354 C-term Y => A N/A N/A Valiquette M et al (1995)
adrb2_human 366 C-term Y => A N/A N/A Valiquette M et al (1995)
adrb2_human 7.39x38 312 TM7 N => F N/A N/A Suryanarayana S et al (1992)
adrb2_human 8.59x59 341 H8 C => G N/A N/A Moffett S et al (1996)
adrb2_human 190 ECL2 C => S N/A N/A Fraser CM et al (1989)
adrb2_human 45.50x50 191 ECL2 C => S N/A N/A Fraser CM et al (1989)
adrb2_human 4.57x57 165 TM4 S => A N/A N/A Wieland K et al (1996)
adrb2_human 6.55x55 293 TM6 N => L N/A N/A Wieland K et al (1996)
adrb2_human 7.53x53 326 TM7 Y => F N/A N/A Gabilondo AM et al (1996)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Gabilondo AM et al (1996)
adrb2_human 413 C-term L => A N/A N/A Hall RA et al (1998)
adrb2_human 412 C-term L => A N/A N/A Hall RA et al (1998)
adrb2_human 411 C-term S => A N/A N/A Hall RA et al (1998)
adrb2_human 410 C-term D => A N/A N/A Hall RA et al (1998)
adrb2_human 7.33x32 306 TM7 E => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.34x33 307 TM7 V => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.35x34 308 TM7 Y => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.36x35 309 TM7 I => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.37x36 310 TM7 L => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.38x37 311 TM7 L => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.41x40 314 TM7 I => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.44x43 317 TM7 V => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.47x47 320 TM7 G => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.51x51 324 TM7 L => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.35x34 308 TM7 Y => A N/A N/A Kurose H et al (1998)
adrb2_human 7.36x35 309 TM7 I => A N/A N/A Kurose H et al (1998)
adrb2_human 8.59x59 341 H8 C => G N/A N/A Hebert TE et al (1998)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Zhang J et al (1997)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Kikkawa H et al (1997)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Kikkawa H et al (1997)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Menard L et al (1997)
adrb2_human 413 C-term L => A N/A N/A Hall RA et al (1998)
adrb2_human 3.35x35 116 TM3 C => F N/A N/A Zuscik MJ et al (1998)
adrb2_human 7.33x32 306 TM7 E => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.34x33 307 TM7 V => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.35x34 308 TM7 Y => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.36x35 309 TM7 I => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.37x36 310 TM7 L => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.38x37 311 TM7 L => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.41x40 314 TM7 I => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.44x43 317 TM7 V => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.47x47 320 TM7 G => A N/A N/A Kikkawa H et al (1998)
adrb2_human 7.51x51 324 TM7 L => A N/A N/A Kikkawa H et al (1998)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Kikkawa H et al (1998)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Kikkawa H et al (1998)
adrb2_human 8.57x57 339 H8 L => A N/A N/A Gabilondo AM et al (1997)
adrb2_human 8.58x58 340 H8 L => A N/A N/A Gabilondo AM et al (1997)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Rasmussen SG et al (1999)
adrb2_human 3.49x49 130 TM3 D => A N/A N/A Rasmussen SG et al (1999)
adrb2_human 6.47x47 285 TM6 C => S N/A N/A Rasmussen SG et al (1999)
adrb2_human 8.59x59 341 H8 C => G N/A N/A Lachance M et al (1999)
adrb2_human 7.39x38 312 TM7 N => H N/A N/A Elling CE et al (1999)
adrb2_human 7.39x38 312 TM7 N => C N/A N/A Elling CE et al (1999)
adrb2_human 3.32x32 113 TM3 D => A N/A N/A Elling CE et al (1999)
adrb2_human 3.32x32 113 TM3 D => C N/A N/A Elling CE et al (1999)
adrb2_human 3.32x32 113 TM3 D => H N/A N/A Elling CE et al (1999)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Rasmussen SG et al (1999)
adrb2_human 3.49x49 130 TM3 D => A N/A N/A Rasmussen SG et al (1999)
adrb2_human 3.49x49 130 TM3 D => A N/A N/A Ghanouni P et al (2000)
adrb2_human 6.30x30 268 TM6 E => A N/A N/A Ghanouni P et al (2000)
adrb2_human 3.41x41 122 TM3 E => A N/A N/A Ghanouni P et al (2000)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Ambrosio C et al (2000)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Ambrosio C et al (2000)
adrb2_human 5.43x44 204 TM5 S => C N/A N/A Ambrosio C et al (2000)
adrb2_human 5.46x461 207 TM5 S => C N/A N/A Ambrosio C et al (2000)
adrb2_human 5.42x43 203 TM5 S => A N/A N/A Sato T et al (1999)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Sato T et al (1999)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Sato T et al (1999)
adrb2_human 6.31x31 269 TM6 H => A N/A N/A Sheikh SP et al (1999)
adrb2_human 6.30x30 268 TM6 E => H N/A N/A Sheikh SP et al (1999)
adrb2_human 6.32x32 270 TM6 K => H N/A N/A Sheikh SP et al (1999)
adrb2_human 6.33x33 271 TM6 A => H N/A N/A Sheikh SP et al (1999)
adrb2_human 6.34x34 272 TM6 L => H N/A N/A Sheikh SP et al (1999)
adrb2_human 6.35x35 273 TM6 K => H N/A N/A Sheikh SP et al (1999)
adrb2_human 3.53x53 134 TM3 A => H N/A N/A Sheikh SP et al (1999)
adrb2_human 5.42x43 203 TM5 S => T N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => C N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => A N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => V N/A N/A Liapakis G et al (2000)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Liapakis G et al (2000)
adrb2_human 2.48x48 77 TM2 C => V N/A N/A Jensen AD et al (2001)
adrb2_human 2.48x48 77 TM2 C => V N/A N/A Javitch JA et al (1997)
adrb2_human 2.48x48 77 TM2 C => V N/A N/A Gether U et al (1997)
adrb2_human 2.50x50 79 TM2 D => N N/A N/A Liapakis G et al (2004)
adrb2_human 2.64x63 93 TM2 H => A N/A N/A Elling CE et al (1999)
adrb2_human 2.64x63 93 TM2 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 3.32x32 113 TM3 D => A N/A N/A Elling CE et al (1999)
adrb2_human 3.32x32 113 TM3 D => H N/A N/A Elling CE et al (1999)
adrb2_human 3.35x35 116 TM3 C => F N/A N/A Zuscik MJ et al (1998)
adrb2_human 3.35x35 116 TM3 C => V N/A N/A Javitch JA et al (1997)
adrb2_human 3.35x35 116 TM3 C => V N/A N/A Gether U et al (1997)
adrb2_human 3.41x41 122 TM3 E => A N/A N/A Ghanouni P et al (2000)
adrb2_human 3.43x43 124 TM3 L => A N/A N/A Tao YX et al (2000)
adrb2_human 3.43x43 124 TM3 L => K N/A N/A Tao YX et al (2000)
adrb2_human 3.43x43 124 TM3 L => R N/A N/A Tao YX et al (2000)
adrb2_human 3.44x44 125 TM3 C => V N/A N/A Javitch JA et al (1997)
adrb2_human 3.44x44 125 TM3 C => V N/A N/A Gether U et al (1997)
adrb2_human 3.49x49 130 TM3 D => A N/A N/A Rasmussen SG et al (1999)
adrb2_human 3.49x49 130 TM3 D => A N/A N/A Ghanouni P et al (2000)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Rasmussen SG et al (1999)
adrb2_human 3.53x53 134 TM3 A => H N/A N/A Sheikh SP et al (1999)
adrb2_human 34.51x51 139 ICL2 F => A N/A N/A Moro O et al (1994)
adrb2_human 4.56x56 164 TM4 T => I N/A N/A Wieland K et al (1996)
adrb2_human 4.57x57 165 TM4 S => A N/A N/A Wieland K et al (1996)
adrb2_human 4.64x64 172 TM4 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 175 ECL2 R => E N/A N/A Gurevich VV et al (1997)
adrb2_human 178 ECL2 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 5.42x43 203 TM5 S => A N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => C N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => T N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => V N/A N/A Liapakis G et al (2000)
adrb2_human 5.42x43 203 TM5 S => X N/A N/A Liapakis G et al (2000)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Liapakis G et al (2000)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Del Carmine R et al (2002)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Liapakis G et al (2000)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Del Carmine R et al (2002)
adrb2_human 5.63x63 224 TM5 Q => K N/A N/A Ghanouni P et al (2001)
adrb2_human 5.64x64 225 TM5 E => A N/A N/A Swaminath G et al (2003)
adrb2_human 241 ICL3 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 256 ICL3 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 261 ICL3 S => A N/A N/A Zamah AM et al (2002)
adrb2_human 261 ICL3 S => D N/A N/A Zamah AM et al (2002)
adrb2_human 6.24x24 262 TM6 S => A N/A N/A Zamah AM et al (2002)
adrb2_human 6.24x24 262 TM6 S => D N/A N/A Zamah AM et al (2002)
adrb2_human 6.27x27 265 TM6 C => A N/A N/A Jensen AD et al (2001)
adrb2_human 6.27x27 265 TM6 C => A N/A N/A Swaminath G et al (2003)
adrb2_human 6.27x27 265 TM6 C => A N/A N/A Gether U et al (1997)
adrb2_human 6.28x28 266 TM6 L => S N/A N/A Rasmussen SG et al (1999)
adrb2_human 6.28x28 266 TM6 L => S N/A N/A Liapakis G et al (2004)
adrb2_human 6.28x28 266 TM6 L => S N/A N/A Javitch JA et al (1997)
adrb2_human 6.29x29 267 TM6 K => R N/A N/A Rasmussen SG et al (1999)
adrb2_human 6.29x29 267 TM6 K => R N/A N/A Liapakis G et al (2004)
adrb2_human 6.29x29 267 TM6 K => R N/A N/A Javitch JA et al (1997)
adrb2_human 6.30x30 268 TM6 E => A N/A N/A Ghanouni P et al (2000)
adrb2_human 6.31x31 269 TM6 H => A N/A N/A Sheikh SP et al (1999)
adrb2_human 6.31x31 269 TM6 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 6.31x31 269 TM6 H => C N/A N/A Jensen AD et al (2001)
adrb2_human 6.31x31 269 TM6 H => K N/A N/A Rasmussen SG et al (1999)
adrb2_human 6.31x31 269 TM6 H => K N/A N/A Liapakis G et al (2004)
adrb2_human 6.31x31 269 TM6 H => K N/A N/A Javitch JA et al (1997)
adrb2_human 6.32x32 270 TM6 K => C N/A N/A Jensen AD et al (2001)
adrb2_human 6.33x33 271 TM6 A => C N/A N/A Jensen AD et al (2001)
adrb2_human 6.34x34 272 TM6 L => A N/A N/A Rasmussen SG et al (1999)
adrb2_human 6.34x34 272 TM6 L => A N/A N/A Liapakis G et al (2004)
adrb2_human 6.34x34 272 TM6 L => A N/A N/A Javitch JA et al (1997)
adrb2_human 6.34x34 272 TM6 L => C N/A N/A Jensen AD et al (2001)
adrb2_human 6.34x34 272 TM6 L => H N/A N/A Sheikh SP et al (1999)
adrb2_human 6.47x47 285 TM6 C => S N/A N/A Rasmussen SG et al (1999)
adrb2_human 6.47x47 285 TM6 C => S N/A N/A Javitch JA et al (1997)
adrb2_human 6.47x47 285 TM6 C => S N/A N/A Gether U et al (1997)
adrb2_human 6.55x55 293 TM6 N => L N/A N/A Wieland K et al (1996)
adrb2_human 6.58x58 296 TM6 H => A N/A N/A Elling CE et al (1999)
adrb2_human 6.58x58 296 TM6 H => A N/A N/A Swaminath G et al (2003)
adrb2_human 7.32x31 305 TM7 K => R N/A N/A Parola AL et al (1997)
adrb2_human 7.37x36 310 TM7 L => F N/A N/A Mizobe T et al (1996)
adrb2_human 7.38x37 311 TM7 L => F N/A N/A Mizobe T et al (1996)
adrb2_human 7.39x38 312 TM7 N => C N/A N/A Elling CE et al (1999)
adrb2_human 7.39x38 312 TM7 N => F N/A N/A Mizobe T et al (1996)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Millman EE et al (2004)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Ferguson SS et al (1995)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Menard L et al (1996)
adrb2_human 7.54x54 327 TM7 C => S N/A N/A Jensen AD et al (2001)
adrb2_human 7.54x54 327 TM7 C => S N/A N/A Javitch JA et al (1997)
adrb2_human 7.54x54 327 TM7 C => S N/A N/A Gether U et al (1997)
adrb2_human 8.56x56 338 H8 E => Q N/A N/A Belanger C et al (2001)
adrb2_human 8.57x57 339 H8 L => A N/A N/A Gabilondo AM et al (1997)
adrb2_human 8.58x58 340 H8 L => A N/A N/A Gabilondo AM et al (1997)
adrb2_human 8.59x59 341 H8 C => G N/A N/A O'Dowd BF et al (1989)
adrb2_human 8.59x59 341 H8 C => G N/A N/A Jin H et al (1997)
adrb2_human 8.59x59 341 H8 C => S N/A N/A Belanger C et al (2001)
adrb2_human 342 C-term L => Y N/A N/A Belanger C et al (2001)
adrb2_human 345 C-term S => A N/A N/A Zamah AM et al (2002)
adrb2_human 345 C-term S => D N/A N/A Zamah AM et al (2002)
adrb2_human 346 C-term S => A N/A N/A Zamah AM et al (2002)
adrb2_human 346 C-term S => A N/A N/A Ferguson SS et al (1995)
adrb2_human 346 C-term S => D N/A N/A Zamah AM et al (2002)
adrb2_human 356 C-term S => G N/A N/A Jockers R et al (1996)
adrb2_human 364 C-term S => A N/A N/A Oakley RH et al (2001)
adrb2_human 364 C-term S => G N/A N/A Jockers R et al (1996)
adrb2_human 378 C-term C => A N/A N/A Jensen AD et al (2001)
adrb2_human 378 C-term C => A N/A N/A Ghanouni P et al (2001)
adrb2_human 378 C-term C => A N/A N/A Gether U et al (1997)
adrb2_human 378 C-term C => V N/A N/A Jensen AD et al (2001)
adrb2_human 406 C-term C => A N/A N/A Jensen AD et al (2001)
adrb2_human 406 C-term C => A N/A N/A Ghanouni P et al (2001)
adrb2_human 406 C-term C => A N/A N/A Gether U et al (1997)
adrb2_human 406 C-term C => V N/A N/A Jensen AD et al (2001)
adrb2_human 407 C-term S => G N/A N/A Ferguson SS et al (1995)
adrb2_human 410 C-term D => A N/A N/A Cong M et al (2001)
adrb2_human 410 C-term D => A N/A N/A Xiang Y et al (2003)
adrb2_human 411 C-term S => A N/A N/A Cong M et al (2001)
adrb2_human 411 C-term S => A N/A N/A Ferguson SS et al (1995)
adrb2_human 412 C-term L => A N/A N/A Cong M et al (2001)
adrb2_human 412 C-term L => A N/A N/A Xiang Y et al (2003)
adrb2_human 413 C-term L => A N/A N/A Maudsley S et al (2000)
adrb2_human 413 C-term L => A N/A N/A Cong M et al (2001)
adrb2_human 413 C-term L => A N/A N/A Naren AP et al (2003)
adrb2_human 7.46x46 319 TM7 S => A N/A N/A Gouldson PR et al (1997)
adrb2_human 7.39x38 312 TM7 N => F N/A N/A Gouldson PR et al (1997)
adrb2_human 7.39x38 312 TM7 N => T N/A N/A Gouldson PR et al (1997)
adrb2_human 7.39x38 312 TM7 N => A N/A N/A Gouldson PR et al (1997)
adrb2_human 6.47x47 285 TM6 C => S N/A N/A Gouldson PR et al (1997)
adrb2_human 6.30x30 268 TM6 E => G N/A N/A Gouldson PR et al (1997)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Gouldson PR et al (1997)
adrb2_human 34.50x50 138 ICL2 P => T N/A N/A Gouldson PR et al (1997)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Gouldson PR et al (1997)
adrb2_human 3.32x32 113 TM3 D => Q N/A N/A Gouldson PR et al (1997)
adrb2_human 2.50x50 79 TM2 D => N N/A N/A Gouldson PR et al (1997)
adrb2_human 2.50x50 79 TM2 D => A N/A N/A Gouldson PR et al (1997)
adrb2_human 12.50x50 64 ICL1 L => K N/A N/A Gouldson PR et al (1997)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Gouldson PR et al (1997)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Kikkawa H et al (1998)
adrb2_human 6.30x30 268 TM6 E => A N/A N/A Ballesteros JA et al (2001)
adrb2_human 6.30x30 268 TM6 E => Q N/A N/A Ballesteros JA et al (2001)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Ballesteros JA et al (2001)
adrb2_human 6.44x44 282 TM6 F => R N/A N/A Rosenbaum DM et al (2011)
adrb2_human 2.64x63 93 TM2 H => C N/A N/A Rosenbaum DM et al (2011)
adrb2_human 187 ECL2 N => E N/A N/A Rosenbaum DM et al (2011)
adrb2_human 3.41x41 122 TM3 E => W N/A N/A Jaakola VP et al (2010)
adrb2_human 6.44x44 282 TM6 F => N N/A N/A Rasmussen SG et al (2011)
adrb2_human 5.46x461 207 TM5 S => A N/A N/A Katritch V et al (2009)
adrb2_human 5.43x44 204 TM5 S => C N/A N/A Deupi X et al (2010)
adrb2_human 5.42x43 203 TM5 S => P N/A N/A Rasmussen SG et al (2011)
adrb2_human 3.40x40 121 TM3 I => P N/A N/A Rasmussen SG et al (2011)
adrb2_human 3.40x40 121 TM3 I => N N/A N/A Rasmussen SG et al (2011)
adrb2_human 7.45x45 318 TM7 N => F N/A N/A Rasmussen SG et al (2011)
adrb2_human 5.50x50 211 TM5 P => F N/A N/A Rasmussen SG et al (2011)
adrb2_human 5.43x44 204 TM5 S => A N/A N/A Katritch V et al (2009)
adrb2_human 7.35x34 308 TM7 Y => A N/A N/A Katritch V et al (2009)
adrb2_human 7.39x38 312 TM7 N => A N/A N/A Katritch V et al (2009)
adrb2_human 7.35x34 308 TM7 Y => F N/A N/A Katritch V et al (2009)
adrb2_human 7.35x34 308 TM7 Y => S N/A N/A Rosenbaum DM et al (2011)
adrb2_human 3.40x40 121 TM3 I => P N/A N/A Rosenbaum DM et al (2011)
adrb2_human 5.50x50 211 TM5 P => I N/A N/A Rosenbaum DM et al (2011)
adrb2_human 3.40x40 121 TM3 I => F N/A N/A Rosenbaum DM et al (2011)
adrb2_human 5.50x50 211 TM5 P => F N/A N/A Rosenbaum DM et al (2011)
adrb2_human 3.49x49 130 TM3 D => N N/A N/A Leach K et al (2011)
adrb2_human 3.41x41 122 TM3 E => W N/A N/A Lebon G et al (2011)
adrb2_human 3.43x43 124 TM3 L => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 6.30x30 268 TM6 E => A N/A N/A Schneider EH et al (2010)
adrb2_human 7.49x49 322 TM7 N => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 4.56x56 164 TM4 T => I N/A N/A Warne T et al (2011)
adrb2_human 6.34x34 272 TM6 L => C N/A N/A Rosenbaum DM et al (2007)
adrb2_human 8.57x57 339 H8 L => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 389 C-term G => A N/A N/A Daly AK et al (2010)
adrb2_human 34.51x51 139 ICL2 F => A N/A N/A Rasmussen SG et al (2011)
adrb2_human 187 ECL2 N => E N/A N/A Rasmussen SG et al (2011)
adrb2_human 251 ICL3 D => V N/A N/A Meletiadis J et al (2006)
adrb2_human 4.56x56 164 TM4 T => I N/A N/A Rosenbaum DM et al (2007)
adrb2_human 7.45x45 318 TM7 N => K N/A N/A Rosenbaum DM et al (2007)
adrb2_human 34.51x51 139 ICL2 F => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 3.35x35 116 TM3 C => F N/A N/A Rosenbaum DM et al (2007)
adrb2_human 187 ECL2 N => E N/A N/A Rosenbaum DM et al (2007)
adrb2_human 8.58x58 340 H8 L => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 3.49x49 130 TM3 D => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 7.50x50 323 TM7 P => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 2.50x50 79 TM2 D => N N/A N/A Rosenbaum DM et al (2007)
adrb2_human 6.47x47 285 TM6 C => T N/A N/A Rosenbaum DM et al (2007)
adrb2_human 7.53x53 326 TM7 Y => A N/A N/A Rosenbaum DM et al (2007)
adrb2_human 3.41x41 122 TM3 E => W N/A N/A Hanson MA et al (2008)
adrb2_human 2.42x42 71 TM2 F => L N/A N/A Brockhoff A et al (2010)
adrb2_human 5.42x43 203 TM5 S => A 1.417↑ K(i) (Binding - Radioligand competition/displacement) DETERENOL Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 1.647↓ K(i) (Binding - Radioligand competition/displacement) DETERENOL Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => A 1.36↑ K(i) (Binding - Radioligand competition/displacement) DETERENOL Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 55.556↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => 3.717↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 7.33x32 306 TM7 E => A 1.093↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.34x33 307 TM7 V => A 1.464↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 16.393↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 4.878↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.37x36 310 TM7 L => A 1.279↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.38x37 311 TM7 L => A 2.793↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.41x40 314 TM7 I => A 1.344↑ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.44x43 317 TM7 V => A 1.372↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.47x47 320 TM7 G => A 2.092↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.51x51 324 TM7 L => A 4.878↓ K(i) (Binding - Radioligand competition/displacement) CARMOTEROL Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => A 1.0 K(d) (Binding - Radioligand saturation) CHEMBL1159723 Rasmussen SG et al (1999) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.1↓ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Rasmussen SG et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.64x64 225 TM5 E => A 1.686↓ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 5.64x64 225 TM5 E => A 3.364↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.27x27 265 TM6 C => A 1.227↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.27x27 265 TM6 C => A 8.81↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.31x31 269 TM6 H => C 1.467↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.31x31 269 TM6 H => A 2.188↓ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.31x31 269 TM6 H => A 3.7↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.32x32 270 TM6 K => C 1.082↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.33x33 271 TM6 A => C 1.179↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.34x34 272 TM6 L => C 1.435↑ K(d) (Binding - Radioligand saturation) CHEMBL1159723 Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.261↑ K(d) (Binding - Radioligand competition/displacement) CHEMBL1159723 Gether U et al (1997) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 26.316↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => 12.5↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.57x57 339 H8 L => A 1.0 K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.57x57 339 H8 L => A 1.109↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.58x58 340 H8 L => A 1.4↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.58x58 340 H8 L => A 1.279↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => V 2.232↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => S 1.133↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 40.0↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.25x25 106 TM3 C => V 27.027↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => V 1.444↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.41x41 122 TM3 E => A 5.747↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 3.41x41 122 TM3 E => A 1.835↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 3.44x44 125 TM3 C => V 3.534↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 7.04↑ K(d) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 12.903↑ K(d) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => A 12.523↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Rasmussen SG et al (1999) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 24.174↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Rasmussen SG et al (1999) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => A 2.952↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => A 1.667↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 4.57x57 165 TM4 S => A 1.474↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 184 ECL2 C => V 13.889↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => V 26.316↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => S 7.752↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => V 22.222↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => S 1000.0↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 13.889↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 33.333↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => A 10.989↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => A 1.771↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => A 2.308↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => V 3.25↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.2↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 8.929↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q 16.129↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T 125.0↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => F 2.591↓ K(h) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => A 1.616↓ K(l) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => F 1.196↓ K(l) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => S 1.8↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 8.57x57 339 H8 L => A 1.167↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.58x58 340 H8 L => A 1.221↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 3.41x41 122 TM3 E => A 4.167↓ K(d) (Binding - Radioligand competition/displacement) CHEMBL1160734 Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => A 3.61↓ K(d) (Binding - Radioligand competition/displacement) CHEMBL1160734 Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => A 3.333↓ K(d) (Binding - Radioligand competition/displacement) CHEMBL1160734 Ghanouni P et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 4.902↓ pK(i) (Binding - Radioligand competition/displacement) phenylephrine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 4.673↓ pK(i) (Binding - Radioligand competition/displacement) phenylephrine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 1.289↓ pK(i) (Binding - Radioligand competition/displacement) phenylephrine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 1.585↓ pK(i) (Binding - Radioligand competition/displacement) phenylephrine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 6.623↓ pK(i) (Binding - Radioligand competition/displacement) phenylephrine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 5.747↓ pK(i) (Binding - Radioligand competition/displacement) (+/-)-Halostachine Liapakis G et al (2004) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 3.89↑ pK(i) (Binding - Radioligand competition/displacement) (+/-)-Halostachine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 1.259↑ pK(i) (Binding - Radioligand competition/displacement) (+/-)-Halostachine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 1.072↓ pK(i) (Binding - Radioligand competition/displacement) (+/-)-Halostachine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 3.802↑ pK(i) (Binding - Radioligand competition/displacement) (+/-)-Halostachine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 4.167↓ pK(i) (Binding - Radioligand competition/displacement) (+/-)-Halostachine Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 3.155↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => 1.522↑ K(i) (Binding - Radioligand competition/displacement) salmeterol Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 7.33x32 306 TM7 E => A 1.996↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.34x33 307 TM7 V => A 1.451↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 111.111↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 111.111↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 15.152↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 11.765↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.37x36 310 TM7 L => A 1.263↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.38x37 311 TM7 L => A 1.009↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.41x40 314 TM7 I => A 1.263↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.44x43 317 TM7 V => A 1.389↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.47x47 320 TM7 G => A 1.894↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.51x51 324 TM7 L => A 2.967↓ K(i) (Binding - Radioligand competition/displacement) salmeterol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.867↑ K(i) (Binding - Radioligand competition/displacement) CHEMBL1396140 Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 250.0↓ K(i) (Binding - Radioligand competition/displacement) (-)-noradrenaline Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 3.982↑ K(d) (Binding - Radioligand competition/displacement) (-)-noradrenaline Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 10.989↓ K(i) (Binding - Radioligand competition/displacement) (-)-noradrenaline Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => A Abolishment K(i) (Binding - Radioligand competition/displacement) yohimbine Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => F Abolishment K(i) (Binding - Radioligand competition/displacement) yohimbine Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q 11.096↑ K(i) (Binding - Radioligand competition/displacement) yohimbine Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T 15.0↑ K(i) (Binding - Radioligand competition/displacement) yohimbine Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 16 N-term G => R 1.131↑ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Green SA et al (1994) Kooistra AJ et al (2013)
adrb2_human 1.26x26 27 TM1 E => N 1.397↑ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Green SA et al (1994) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => V 3.058↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 71.429↓ pK(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Liapakis G et al (2004) Kooistra AJ et al (2013)
adrb2_human 3.25x25 106 TM3 C => V 1000.0↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => V 1.2↑ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 50.0↑ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 3.44x44 125 TM3 C => V 11.364↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 3.937↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 184 ECL2 C => V 43.478↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => V 142.857↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => V 166.667↓ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 25.0↓ pK(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 71.429↓ pK(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 2.755↓ pK(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 40.0↓ pK(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 33.333↓ pK(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => V 3.789↑ K(i) (Binding - Radioligand competition/displacement) (±)-adrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.536↓ K(i) (Binding - Radioligand competition/displacement) terbutaline Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 5.917↓ K(i) (Binding - Radioligand competition/displacement) CHEMBL1800935 Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 15.385↓ K(i) (Binding - Radioligand competition/displacement) CHEMBL1800935 Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 4.608↓ K(i) (Binding - Radioligand competition/displacement) L-NOREPINEPHRINE Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 1.047↓ K(i) (Binding - Radioligand competition/displacement) CHEMBL210309 Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 3.663↓ K(i) (Binding - Radioligand competition/displacement) alprenolol Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 1.637↓ K(i) (Binding - Radioligand competition/displacement) alprenolol Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 1.445↑ pK(i) (Binding - Radioligand competition/displacement) alprenolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 2.041↓ pK(i) (Binding - Radioligand competition/displacement) alprenolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 2.188↓ pK(i) (Binding - Radioligand competition/displacement) alprenolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 1.072↑ pK(i) (Binding - Radioligand competition/displacement) alprenolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => A Abolishment K(i) (Binding - Radioligand competition/displacement) alprenolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q 8.696↓ K(i) (Binding - Radioligand competition/displacement) alprenolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T 111.111↓ K(i) (Binding - Radioligand competition/displacement) alprenolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 1.862↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 3.333↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 11.22↑ pK(i) (Binding - Radioligand competition/displacement) (-)-propranolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 5.37↑ pK(i) (Binding - Radioligand competition/displacement) (-)-propranolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 1.38↑ pK(i) (Binding - Radioligand competition/displacement) (-)-propranolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 2.239↑ pK(i) (Binding - Radioligand competition/displacement) (-)-propranolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => S 1.259↓ K(i) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 1.0 K(i) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.767↓ K(d) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => S 76.923↓ K(i) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => S 250.0↓ K(i) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.259↑ K(i) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => S 1.0 K(i) (Binding - Radioligand competition/displacement) DEXPROPRANOLOL Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 5.917↓ K(i) (Binding - Radioligand competition/displacement) CGP 20712A Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 18.28↑ K(i) (Binding - Radioligand competition/displacement) DICHLOROISOPROTERENOL Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 8.13↓ pK(i) (Binding - Radioligand competition/displacement) DEOXIEPINEPHRINE Liapakis G et al (2004) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 3.774↓ K(i) (Binding - Radioligand competition/displacement) METATEROL Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 6.711↓ K(i) (Binding - Radioligand competition/displacement) METATEROL Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => A 1.571↑ K(i) (Binding - Radioligand competition/displacement) METATEROL Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 4.467↑ pK(i) (Binding - Radioligand competition/displacement) OXEDRINE Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 2.818↑ pK(i) (Binding - Radioligand competition/displacement) OXEDRINE Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 1.38↑ pK(i) (Binding - Radioligand competition/displacement) OXEDRINE Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 3.467↑ pK(i) (Binding - Radioligand competition/displacement) OXEDRINE Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 1.023↑ pK(i) (Binding - Radioligand competition/displacement) OXEDRINE Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.233↓ K(d) (Binding - Radioligand saturation) CGP 12177 Shi L et al (2002) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => T 1.11↓ K(d) (Binding - Radioligand saturation) CGP 12177 Shi L et al (2002) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 7.949↑ K(i) (Binding - Radioligand competition/displacement) CGP 12177 Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.0 K(i) (Binding - Radioligand competition/displacement) CGP 12177 Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 1.057↑ K(i) (Binding - Radioligand competition/displacement) CGP 12177 Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 3.472↓ pK(i) (Binding - Radioligand competition/displacement) CGP 12177 Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 9.524↓ pK(i) (Binding - Radioligand competition/displacement) CGP 12177 Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 1.698↑ pK(i) (Binding - Radioligand competition/displacement) CGP 12177 Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 6.452↓ pK(i) (Binding - Radioligand competition/displacement) CGP 12177 Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => A 2.331↓ K(i) (Binding - Radioligand competition/displacement) CGP 12177 Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => Q 2.0↓ K(i) (Binding - Radioligand competition/displacement) CGP 12177 Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 6.667↑ K(d) (Binding - Radioligand competition/displacement) (+)-adrenaline Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 14.706↓ K(i) (Binding - Radioligand competition/displacement) (+)-adrenaline Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => V 3.968↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 15.385↓ pK(i) (Binding - Radioligand competition/displacement) noradrenaline Liapakis G et al (2004) Kooistra AJ et al (2013)
adrb2_human 3.25x25 106 TM3 C => V 18.868↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => V 1.381↑ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.44x44 125 TM3 C => V 4.651↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 4.329↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 184 ECL2 C => V 55.556↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => V 22.222↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => V 20.833↓ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => V 2.417↑ K(i) (Binding - Radioligand competition/displacement) noradrenaline Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 16 N-term G => R 1.25↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Green SA et al (1994) Kooistra AJ et al (2013)
adrb2_human 1.26x26 27 TM1 E => N 1.56↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Green SA et al (1994) Kooistra AJ et al (2013)
adrb2_human 12.50x50 64 ICL1 L => G 10.801↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 75.0↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 113.035↑ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 34.50x50 138 ICL2 P => T 1.04↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 34.50x50 138 ICL2 P => T 1.031↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 4.329↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 25.0↓ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ambrosio C et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => C 31.25↓ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ambrosio C et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => A 15.873↓ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ambrosio C et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => A 20.0↓ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ambrosio C et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.64x64 225 TM5 E => A 1.209↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 5.64x64 225 TM5 E => A 1.89↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.27x27 265 TM6 C => A 1.833↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.27x27 265 TM6 C => A 2.16↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => G 4.57↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => A 2.812↑ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => Q 1.406↑ K(d) (Binding - Radioligand competition/displacement) isoprenaline Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.31x31 269 TM6 H => C 1.6↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.31x31 269 TM6 H => A 2.0↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.31x31 269 TM6 H => A 6.494↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Swaminath G et al (2003) Kooistra AJ et al (2013)
adrb2_human 6.32x32 270 TM6 K => C 1.6↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.33x33 271 TM6 A => C 2.192↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.34x34 272 TM6 L => C 3.721↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Jensen AD et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.188↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Gether U et al (1997) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 2.049↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Shi L et al (2002) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => T 5.167↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Shi L et al (2002) Kooistra AJ et al (2013)
adrb2_human 7.33x32 306 TM7 E => A 1.2↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.34x33 307 TM7 V => A 1.376↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 5.405↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 1.499↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.37x36 310 TM7 L => A 1.167↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.38x37 311 TM7 L => A 1.499↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.41x40 314 TM7 I => A 1.6↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.44x43 317 TM7 V => A 1.292↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.47x47 320 TM7 G => A 2.0↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.49x49 322 TM7 N => A 3.425↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.49x49 322 TM7 N => D 1.479↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.49x49 322 TM7 N => D 1.381↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.50x50 323 TM7 P => A 4.808↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.50x50 323 TM7 P => A 2.283↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.51x51 324 TM7 L => A 1.167↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => F 5.988↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => F 2.717↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1995) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => A 20.5↑ K(h) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1994) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => A 3.486↑ K(l) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1994) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => A 1.159↑ K(l) (Binding - Radioligand competition/displacement) isoprenaline Barak LS et al (1994) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => R 3.125↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => R 3.846↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 1.114↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1989) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 1.087↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 1.04↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline O'Dowd BF et al (1988) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 1.232↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Moffett S et al (1993) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 2.212↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Moffett S et al (1996) Kooistra AJ et al (2013)
adrb2_human 350 C-term Y => A 4.75↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Valiquette M et al (1993) Kooistra AJ et al (2013)
adrb2_human 350 C-term Y => A 1.304↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Valiquette M et al (1993) Kooistra AJ et al (2013)
adrb2_human 354 C-term Y => A 4.184↓ K(i) (Binding - Radioligand competition/displacement) isoprenaline Valiquette M et al (1993) Kooistra AJ et al (2013)
adrb2_human 354 C-term Y => A 2.582↑ K(i) (Binding - Radioligand competition/displacement) isoprenaline Valiquette M et al (1993) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => S 1.585↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 1.0 K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.637↓ K(d) (Binding - Radioligand competition/displacement) (-)-propranolol Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => S 100.0↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => S N/A K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.259↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q 20.0↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T 1000.0↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => S 1.259↓ K(i) (Binding - Radioligand competition/displacement) (-)-propranolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => V 1.733↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => S 1.0 K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 62.5↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.25x25 106 TM3 C => V 52.632↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => V 1.659↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.44x44 125 TM3 C => V 4.016↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 6.154↑ K(d) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 4.57x57 165 TM4 S => A 3.759↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 184 ECL2 C => V 13.889↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => V 38.462↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => S 100.0↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => V 166.667↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => S 250.0↓ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => V 1.896↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.0 K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.828↑ K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => S N/A K(i) (Binding - Radioligand competition/displacement) LEVISOPRENALINE Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.042↓ K(i) (Binding - Radioligand competition/displacement) clenbuterol Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 26.316↓ K(i) (Binding - Radioligand competition/displacement) pindolol Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => A 1.12↑ K(i) (Binding - Radioligand competition/displacement) pindolol Rasmussen SG et al (1999) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.011↑ K(i) (Binding - Radioligand competition/displacement) pindolol Rasmussen SG et al (1999) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.835↓ K(i) (Binding - Radioligand competition/displacement) pindolol Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 1.35↓ K(i) (Binding - Radioligand competition/displacement) pindolol Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 24.39↓ pK(i) (Binding - Radioligand competition/displacement) pindolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => C 66.667↓ pK(i) (Binding - Radioligand competition/displacement) pindolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => T 5.128↓ pK(i) (Binding - Radioligand competition/displacement) pindolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => V 66.667↓ pK(i) (Binding - Radioligand competition/displacement) pindolol Liapakis G et al (2000) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => A 3.333↓ K(i) (Binding - Radioligand competition/displacement) pindolol Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 6.30x30 268 TM6 E => Q 5.988↓ K(i) (Binding - Radioligand competition/displacement) pindolol Ballesteros JA et al (2001) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q 1.585↑ K(i) (Binding - Radioligand competition/displacement) pindolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T 50.0↓ K(i) (Binding - Radioligand competition/displacement) pindolol Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 40.0↓ K(i) (Binding - Radioligand competition/displacement) ICI-118551 Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 4.587↓ K(i) (Binding - Radioligand competition/displacement) ICI-118551 Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 1.139↓ K(i) (Binding - Radioligand competition/displacement) dopamine Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.376↓ K(i) (Binding - Radioligand competition/displacement) dopamine Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q Gain of effect (wt had no effect) K(i) (Binding - Radioligand competition/displacement) apraclonidine Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T No effect K(i) (Binding - Radioligand competition/displacement) apraclonidine Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 2.50x50 79 TM2 D => N 142.857↓ K(i) (Binding - Radioligand competition/displacement) (-)-adrenaline Chung FZ et al (1988) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 13.14↑ K(d) (Binding - Radioligand competition/displacement) (-)-adrenaline Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 37.037↓ K(i) (Binding - Radioligand competition/displacement) (-)-adrenaline Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => Q 29.412↓ K(i) (Binding - Radioligand competition/displacement) (-)-adrenaline Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 7.39x38 312 TM7 N => T 5.263↓ K(i) (Binding - Radioligand competition/displacement) (-)-adrenaline Suryanarayana S et al (1993) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 1.5↑ K(i) (Binding - Radioligand competition/displacement) salbutamol Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 2.421↓ K(i) (Binding - Radioligand competition/displacement) salbutamol Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => 1.295↑ K(i) (Binding - Radioligand competition/displacement) salbutamol Kikkawa H et al (1997) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => F 7.059↑ K(i) (Binding - Radioligand competition/displacement) orciprenaline Zuscik MJ et al (1998) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.048↑ K(i) (Binding - Radioligand competition/displacement) dobutamine Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 4.56x56 164 TM4 T => I 1.938↓ K(i) (Binding - Radioligand competition/displacement) dobutamine Green SA et al (1993) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 1.364↓ K(i) (Binding - Radioligand competition/displacement) Iodocyanopindolol Moffett S et al (1996) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => V 1.182↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 2.48x48 77 TM2 C => S 1.259↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 3.25x25 106 TM3 C => V 15.625↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.35x35 116 TM3 C => V 2.273↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.44x44 125 TM3 C => V 1.0 K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 3.49x49 130 TM3 D => N 1.524↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Fraser CM et al (1988) Kooistra AJ et al (2013)
adrb2_human 4.57x57 165 TM4 S => A 1.773↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 184 ECL2 C => V 4.274↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => V 11.236↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 190 ECL2 C => S 2.513↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => V 15.152↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 45.50x50 191 ECL2 C => S 6.329↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 5.42x43 203 TM5 S => A 1.89↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.43x44 204 TM5 S => A 1.363↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 5.46x461 207 TM5 S => A 1.208↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Sato T et al (1999) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => V 1.727↓ K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Dohlman HG et al (1990) Kooistra AJ et al (2013)
adrb2_human 6.47x47 285 TM6 C => S 1.0 K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 6.55x55 293 TM6 N => L 1.119↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Wieland K et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.33x32 306 TM7 E => A 1.065↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.33x32 306 TM7 E => A 1.04↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.34x33 307 TM7 V => A 1.129↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.34x33 307 TM7 V => A 1.018↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 1.148↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 1.043↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 1.047↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 1.096↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 1.147↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 1.089↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.37x36 310 TM7 L => A 1.258↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.37x36 310 TM7 L => A 1.107↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.38x37 311 TM7 L => A 1.107↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.38x37 311 TM7 L => A 1.125↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.41x40 314 TM7 I => A 1.107↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.41x40 314 TM7 I => A 1.079↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.44x43 317 TM7 V => A 1.032↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.44x43 317 TM7 V => A 1.112↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.47x47 320 TM7 G => A 1.58↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.47x47 320 TM7 G => A 1.927↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.51x51 324 TM7 L => A 1.161↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Kikkawa H et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.51x51 324 TM7 L => A 1.418↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => A 1.02↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Gabilondo AM et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.53x53 326 TM7 Y => F 1.112↓ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Gabilondo AM et al (1996) Kooistra AJ et al (2013)
adrb2_human 7.54x54 327 TM7 C => S 1.0 K(i) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Fraser CM et al (1989) Kooistra AJ et al (2013)
adrb2_human 8.57x57 339 H8 L => A 1.014↑ K(d) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.57x57 339 H8 L => A 1.014↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.58x58 340 H8 L => A 1.044↑ K(d) (Binding - Radioligand competition/displacement) [125I]iodocyanopindolol Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.58x58 340 H8 L => A 1.044↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol Gabilondo AM et al (1997) Kooistra AJ et al (2013)
adrb2_human 8.59x59 341 H8 C => G 1.197↑ K(d) (Binding - Radioligand saturation) [125I]iodocyanopindolol O'Dowd BF et al (1989) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 14.493↓ K(i) (Binding - Radioligand competition/displacement) Salmeterol-derivative 2 Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 2.924↓ K(i) (Binding - Radioligand competition/displacement) Salmeterol-derivative 2 Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.35x34 308 TM7 Y => A 10.87↓ K(i) (Binding - Radioligand competition/displacement) Salmeterol-derivative 1 Isogaya M et al (1998) Kooistra AJ et al (2013)
adrb2_human 7.36x35 309 TM7 I => A 2.653↓ K(i) (Binding - Radioligand competition/displacement) Salmeterol-derivative 1 Isogaya M et al (1998) Kooistra AJ et al (2013)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 E R L Q ICL1ECL1 M W T F ECL1ICL2 P F K Y Q S L L ICL2ECL2 W Y R A T H Q E A I N C Y A N E T C C D F F T ECL2ICL3 G R F H V Q N L S Q V E Q D G R T G H G L R R S ICL3ECL3 D N L I ECL3N-term M G Q P G N G S A F L L A P N G S H A P D H D V T N-termC-term L R R S S L K A Y G N G Y S S N G N T G E Q S G Y H V E Q E K E N K L L C E D L P G T E D F V G H Q G T V P S D N I D S Q G R N C S T N D S L L C-term Q E R D E V W V V G M G I V M S L I V L A I V F G N V L V I T A I A K F T V T N Y F I T S L A C A D L V M G L A V V P F G A A H I L M K G N F W C E F W T S I D V L C V T A S I E T L C V I A V D R Y F A I T S T K N K A R V I I L M V W I V S G L T S F L P I Q M H N Q A Y A I A S S I V S F Y V P L V I M V F V Y S R V F Q E A K R Q L Q K I D K S E S K F C L K E H K A L K T L G I I M G T F T L C W L P F F I V N I V H V I Q R K E V Y I L L N W I G Y V N S G F N P L I Y C R S P D F Q E F R I A L L C
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
V N G F V I A L V I L S M V I G M G V V 1 T S L A C A D L V M G A L V V P F G A A H 2 V C L T E I S A T V C L V D I S T W F E 3 A R V I I L M V W I V S G L T S F L P I 4 Y V F V M I V L P V Y F S V I S S A I A Y 5 G I I M G T F T L C W L P F F I V N I V 6 L P N F G S N V Y G I W N L L I Y V E 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
β2-adrenoceptor
TM1
1x26 1.26x26 E27
TM2
2x42 2.42x42 F71
2x48 2.48x48 C77
2x50 2.50x50 D79
2x63 2.64x63 H93
TM3
3x25 3.25x25 C106
3x32 3.32x32 D113
3x35 3.35x35 C116
3x40 3.40x40 I121
3x41 3.41x41 E122
3x43 3.43x43 L124
3x44 3.44x44 C125
3x49 3.49x49 D130
3x53 3.53x53 A134
TM4
4x56 4.56x56 T164
4x57 4.57x57 S165
4x64 4.64x64 H172
TM5
5x43 5.42x43 S203
5x44 5.43x44 S204
5x461 5.46x461 S207
5x50 5.50x50 P211
5x63 5.63x63 Q224
5x64 5.64x64 E225
TM6
6x24 6.24x24 S262
6x27 6.27x27 C265
6x28 6.28x28 L266
6x29 6.29x29 K267
6x30 6.30x30 E268
6x31 6.31x31 H269
6x32 6.32x32 K270
6x33 6.33x33 A271
6x34 6.34x34 L272
6x35 6.35x35 K273
6x44 6.44x44 F282
6x47 6.47x47 C285
6x55 6.55x55 N293
6x58 6.58x58 H296
TM7
7x31 7.32x31 K305
7x32 7.33x32 E306
7x33 7.34x33 V307
7x34 7.35x34 Y308
7x35 7.36x35 I309
7x36 7.37x36 L310
7x37 7.38x37 L311
7x38 7.39x38 N312
7x40 7.41x40 I314
7x43 7.44x43 V317
7x45 7.45x45 N318
7x46 7.46x46 S319
7x47 7.47x47 G320
7x49 7.49x49 N322
7x50 7.50x50 P323
7x51 7.51x51 L324
7x53 7.53x53 Y326
7x54 7.54x54 C327
H8
8x56 8.56x56 E338
8x57 8.57x57 L339
8x58 8.58x58 L340
8x59 8.59x59 C341