Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
cckar_rat 5.74x74 260 TM5 S => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 264 ICL3 S => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 275 ICL3 S => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 424 C-term T => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 7.53x53 386 TM7 Y => A N/A N/A Go WY et al (1998)
cckar_rat 5.67x67 253 TM5 Q => L N/A N/A Silvente-Poirot S et al (1996)
cckar_rat 45.52x52 213 ECL2 F => A N/A N/A Silvente-Poirot S et al (1998)
cckar_rat 2.65x64 117 TM2 N => A N/A N/A Silvente-Poirot S et al (1998)
cckar_rat 2.66x65 118 TM2 L => A N/A N/A Silvente-Poirot S et al (1998)
cckar_rat 23.50x50 122 ECL1 F => A N/A N/A Silvente-Poirot S et al (1998)
cckar_rat 23.52x52 124 ECL1 F => A N/A N/A Silvente-Poirot S et al (1998)
cckar_rat 2.67x66 119 TM2 L => M N/A N/A Dong M et al (2005)
cckar_rat 3.26x26 130 TM3 K => A N/A N/A Gouldson P et al (1999)
cckar_rat 202 ECL2 K => A N/A N/A Gouldson P et al (1999)
cckar_rat 5.74x74 260 TM5 S => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 264 ICL3 S => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 275 ICL3 S => A N/A N/A Ozcelebi F et al (1996)
cckar_rat 360 ECL3 E => G N/A N/A Archer-Lahlou E et al (2005)
cckar_rat 424 C-term T => A N/A N/A Ozcelebi F et al (1996)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 K R M R ICL1ECL1 D F I F ECL1ICL2 P L Q S R V W Q ICL2ECL2 N L V P F T K N N N Q T A N M C R F L L P ECL2ICL3 Q K K S A K E K K P S T G S S T R Y E D S D G C Y L Q K S R P P R K L E L Q Q L S S G S G G S R L N R I R S S S ICL3ECL3 T V S A E K H L S ECL3N-term M S H S P A R Q H L V E S S R M D V V D S L L M N G S N I T P P C E L G L E N E T L F C L D Q P Q P S K E N-termC-term P G P P G V R G E V G E E E D G R T I R A L L S R Y S Y S H M S T S A P P P C-term W Q S A L Q I L L Y S I I F L L S V L G N T L V I T V L I R N T V T N I F L L S L A V S D L M L C L F C M P F N L I P N L L K G S A V C K T T T Y F M G T S V S V S T F N L V A I S L E R Y G A I C R T K S H A L K V I A A T W C L S F T I M T P Y P I Y S S D A M Q Q S W Q T F L L L I L F L L P G I V M V V A Y G L I S L E L Y Q G I K F D A S S A A N L I A K K R V I R M L I V I V V L F F L C W M P I F S A N A W R A Y D G T P I S F I L L L S Y T S S C V N P I I Y C F M N K R F M A C P N F R L G T F P C
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
T N G L V S L L F I I S Y L L I Q L A S 1 L S L A V S D L M L C F L C M P F N L I P 2 A V L N F T S V S V S T G M F Y T T T K 3 A L K V I A A T W C L S F T I M T P Y 4 Y A V V M V I G P L L F L I L L L F T Q W 5 I V I V V L F F L C W M P I F S A N A W 6 I P N V C S S T Y S L L L I F S I P T 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
CCK1 receptor
TM2
2x64 2.65x64 N117
2x65 2.66x65 L118
2x66 2.67x66 L119
TM3
3x26 3.26x26 K130
TM5
5x67 5.67x67 Q253
5x74 5.74x74 S260
TM7
7x53 7.53x53 Y386