Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
cltr1_human 3.35x35 106 TM3 N => A N/A N/A Dupre DJ et al (2004)
cltr1_human 6.34x35 232 TM6 I => R N/A N/A Dupre DJ et al (2004)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 Y H K K ICL1ECL1 G I W L F ECL1ICL2 P V Q N I N L V ICL2ECL2 K P Q K D E K N N T K C F E P P Q ECL2ICL3 K S M K K ICL3ECL3 E T K ECL3N-term M D E T G N L T V S N-termC-term H S L S S V T Y V P R K K A S L P E K G E E I C K V C-term S A T C H D T I D D F R N Q V Y S T L Y S M I S V V G F F G N G F V L Y V L I K T S A F Q V Y M I N L A V A D L L C V C T L P L R V V Y Y V H K G D F L C R L S T Y A L Y V N L Y C S I F F M T A M S F F R C I A I V F T Q K K A R F V C V G I W I F V I L T S S P F L M A D N Q T K N H V L V L H Y V S L F V G F I I P F V I I I V C Y T M I I L T L L K N L S S H K K A I G M I M V V T A A F L V S F M P Y H I Q R T I H L H F L H N P C D S V L R M Q K S V V I T L S L A A S N C C F D P L L Y F F S G G N L S T F R K R F R K
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
G N G F F G V V S I M S Y L T S Y V Q N 1 I N L A V A D L L C V C T L P L R V V Y 2 A T M F F I S C Y L N V Y L A Y T S L R 3 A R F V C V G I W I F V I L T S S P F 4 Y C V I I I V F P I I F G V F L S V Y H L 5 I M V V T A A F V L S F M P Y H I Q R T I 6 L P D F C C N S A A L S L T I V V S K 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
CysLT1 receptor
TM3
3x35 3.35x35 N106
TM6
6x35 6.34x35 I232