Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
opsr_human 1.44x44 65 TM1 T => I N/A N/A Asenjo AB et al (1994)
opsr_human 5.49x49 230 TM5 I => T N/A N/A Asenjo AB et al (1994)
opsr_human 5.52x52 233 TM5 A => S N/A N/A Asenjo AB et al (1994)
opsr_human 6.44x44 277 TM6 Y => F N/A N/A Asenjo AB et al (1994)
opsr_human 6.52x52 285 TM6 T => A N/A N/A Asenjo AB et al (1994)
opsr_human 7.40x39 309 TM7 Y => F N/A N/A Asenjo AB et al (1994)
opsr_human 1.44x44 65 TM1 T => I N/A N/A Merbs SL et al (1993)
opsr_human 5.49x49 230 TM5 I => T N/A N/A Merbs SL et al (1993)
opsr_human 5.52x52 233 TM5 A => S N/A N/A Merbs SL et al (1993)
opsr_human 6.44x44 277 TM6 Y => F N/A N/A Merbs SL et al (1993)
opsr_human 6.52x52 285 TM6 T => A N/A N/A Merbs SL et al (1993)
opsr_human 4.50x50 177 TM4 W => R N/A N/A Gardner JC et al (2010)
opsr_human 4.50x50 177 TM4 W => F N/A N/A Gardner JC et al (2010)
opsr_human 5.55x55 236 TM5 M => V N/A N/A Gardner JC et al (2010)
opsr_human 4.50x50 177 TM4 W => Y N/A N/A Gardner JC et al (2010)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 K K L R ICL1ECL1 Y F V L ECL1ICL2 P F G N V R F ICL2ECL2 W S R Y W P H G L K T S C G P D V F S G S S Y P ECL2ICL3 K E ICL3ECL3 G Y A F ECL3N-term M A Q Q W S L Q R L A G R H P Q D S Y E D S T Q S S I F T Y T N S N S T R G P F E G P N Y H I A N-termC-term K K V D D G S E L S S A S K T E V S S V S S V S P A C-term P R W V Y H L T S V W M I F V V T A S V F T N G L V L A A T M K F H P L N W I L V N L A V A D L A E T V I A S T I S I V N Q V S G G H P M C V L E G Y T V S L C G I T G L W S L A I I S W E R W M V V C K D A K L A I V G I A F S W I W A A V W T A P P I F G G V Q S Y M I V L M V T C C I I P L A I I M L C Y L Q V W L A I R A V A K Q Q S E S T Q K A E K E V T R M V V V M I F A Y C V C W G P Y T F F A C F A A A N P H P L M A A L P A Y F A K S A T I Y N P V I Y V F M N R Q I L Q F R N C L F G
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
G N T F V S A T V V F I M W V S T L H Y 1 V N L A V A D L A E T V I A S T I S I V 2 I A L S W L G T I G C L S V T Y G E L V 3 A I V G I A F S W I W A A V W T A P P I 4 Y C L M I I A L P I I C C T V M L V I M Y 5 V V M I F A Y C V C W G P Y T F F A C F 6 V P N Y I T A S K A F Y A P L A A M L 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
OPN1LW
TM1
1x44 1.44x44 T65
TM4
4x50 4.50x50 W177
TM5
5x49 5.49x49 I230
5x52 5.52x52 A233
5x55 5.55x55 M236
TM6
6x44 6.44x44 Y277
6x52 6.52x52 T285
TM7
7x39 7.40x39 Y309