Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
par3_human 3.47x47 188 TM3 S => A N/A N/A Dong JM et al (1998)
par3_human 238 ECL2 V => L N/A N/A Schmidt VA et al (1996)
par3_human 239 ECL2 Q => A N/A N/A De Cristofaro R et al (2001)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 T R S ICL1ECL1 G N N W V F ECL1ICL2 P F T Y R G L P ICL2ECL2 L K Q E Y Y L V Q P D I T T C H D V H N T C E S S S P F ECL2ICL3 D H R ICL3ECL3 Y Y N N T D G ECL3N-term M K A L I F A A A G L L L L L P T F C Q S G M E N D T N N L A K P T L P I K T F R G A P P N S F E E F P F S A L E G W T G A T I T V K I K C P E E S A S H L H V K N A T M G Y L T N-termC-term S K T R N H S T A Y L T K C-term S S L S T K L I P A I Y L L V F V V G V P A N A V T L W M L F F R I C T T V F Y T N L A I A D F L F C V T L P F K I A Y H L N G E V L C R A T T V I F Y G N M Y C S I L L L A C I S I N R Y L A I V H K H T Y A L V T C G L V W A T V F L Y M L P F F I Q L Y Y F I S L A F F G F L I P F V L I I Y C Y A A I I R T L N A Y W L W Y V K A S L L I L V I F T I C F A P S N I I L I I H H A N Y L Y F I Y L I A L C L G S L N S C L D P F L Y F L M
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
A N A P V G V V F V L L Y I A P I L K T 1 T N L A I A D F L F C V T L P F K I A Y 2 C A L L L I S C Y M N G Y F I V T T A R 3 A L V T C G L V W A T V F L Y M L P F 4 Y C Y I I L V F P I L F G F F A L S I F Y 5 S L L I L V I F I T C F A P S N I I L I I 6 F P D L C S N L S G L C L A I L Y I F 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
PAR3
TM3
3x47 3.47x47 S188